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Carboxymethylated pyridoindole antioxidants as aldose reductase inhibitors: synthesis, activity, partitioning, and molecular modeling
Title Carboxymethylated pyridoindole antioxidants as aldose reductase inhibitors: synthesis, activity, partitioning, and molecular modeling Author Štefek Milan 1950-2023 SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV SCOPUS ORCID Co-authors Šnirc Vladimír 1966-2011 SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV SCOPUS Djoubissie Paul-Omer 1971- SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV SCOPUS Májeková Magdaléna 1958- SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV SCOPUS RID ORCID Demopoulos Vassilis J. Račková Lucia 1975- SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV SCOPUS Bezáková Želmíra Karasu Çimen Carbone Vincenzo El-Kabbani Ossama Source document Bioorganic & medicinal chemistry. Vol.16, no. 9 (2008), p. 4908-4920 Language eng - English Country GB - Great Britian Document kind rozpis článkov z periodík (rbx) Citations TOYOOKA, N. - TAKEDA, D. - MINOSHIMA, Y. - KATO, A. - ADACHI, I. Design, synthesis, and biological effect of (1-OXO-1,2,3,4-TETRAHYDRO-beta-CARBOLIN-9-YL)acetic acids as inhibitor of aldose reductase 2. In HETEROCYCLES. ISSN 0385-5414, 2009, vol. 79, p. 1073-1080. PANTELEON, V. - KOSTAKIS, I.K. - MARAKOS, P. - POULI, N. - ANDREADOU, I. Synthesis and free radical scavenging activity of some new spiropyranocoumarins. In BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. ISSN 0960-894X, 2008, vol. 18, no. 21, p. 5781-5784. DAS-EVCIMEN, N. - YILDIRIM, O. - SUZEN, S. Relationship between aldose reductase and superoxide dismutase inhibition capacities of indole based analogs of melatonin derivatives. In ARCHIVES OF BIOLOGICAL SCIENCES. ISSN 0354-4664, 2009, vol. 61, no. 4, p. 675-681. CALDERONE, V. - TESTAI, L. - MARTELLI, A. - LA MOTTA, C. - SARTINI, S. - DA SETTIMO, F. - BRESCHI, M.C. Anti-ischaemic activity of an antioxidant aldose reductase inhibitor on diabetic and non-diabetic rat hearts. In JOURNAL OF PHARMACY AND PHARMACOLOGY. ISSN 0022-3573, 2010, vol. 62, no. 1, p. 107-113. ALEKSEVEV, R.S. - KURKIN, A.V. - YUROVSKAYA, M.A. Gamma-carbolines and their hydrogenated derivatives. 3. Hydrogenated gamma-carboline derivatives: chemical and biological poperties (review). In Khimiya Geterotsiklicheskikh Soedinenii. ISSN 0132-6244, 2010, no. 10, p. 1447-1484 ENDO, S. - MATSUNAGA, T. - SODA, M. - TAJIMA, K. - ZHAO, H.T. - EL-KABBANI, O. - HARA, A. Selective Inhibition of the Tumor Marker AKR1B10 by Antiinflammatory N-Phenylanthranilic Acids and Glycyrrhetic Acid. In BIOLOGICAL & PHARMACEUTICAL BULLETIN. ISSN 0918-6158, 2010, vol. 33, no. 5, p. 886-890. ALEKSEYEV, R.S. - KURKIN, A.V. - YUROVSKAYA, M.A. Gamma-carbolines and their hydrogenated derivatives 3.* Hydrogenated derivatives of Gamma-carbolines: chemical and biological poperties (review). In CHEMISTRY OF HETEROCYCLIC COMPOUNDS. ISSN 0009-3122, 2011, vol. 46, no. 10, p. 1169-1198. DAS-EVCIMEN, N. - SARIKAYA, M. - KARAASLAN, C.- YILMAZ, A.D. - SHIRINZADEH, H. - SUZEN, S. Rat lung aldose reductase inhibition capacity of substituted Indole Hydrazide/Hydrazone derivatives. In FABAD JOURNAL OF PHARMACEUTICAL SCIENCES. ISSN 1300-4182, 2012, vol. 37, no. 4, p. 169-174 OLGEN, S. - BAKAR, F. - AYDIN, S. - NEBIOGLU, D. - NEBIOGLU, S. Synthesis of new indole-2-carboxamide and 3-acetamide derivatives and evaluation their antioxidant properties. In JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY. ISSN 1475-6366, 2013, vol. 28, no. 1, p. 58-64. IQBAL, Z. - ALI, S. - IQBAL, J. - ABBAS, Q. - QURESHI, I.Z. - HAMEED, S. Dual action spirobicycloimidazolidine-2,4-diones: Antidiabetic agents and inhibitors of aldose reductase-an enzyme involved in diabetic complications. In BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. ISSN 0960-894X, 2013, vol. 23, no. 2, p. 488-491. WANG, L. - GU, Q. - ZHENG, X. - YE, J. - LIU, Z. - LI, J. - HU, X. - HAGLER, A. - XU, J. Discovery of new selective human aldose reductase inhibitors through virtual screening multiple binding pocket conformations. In JOURNAL OF CHEMICAL INFORMATION AND MODELING. ISSN 1549-9596, 2013, vol. 53, no. 9, p. 2409-2422 KAUR, A. - SINGH, B. - VYAS, B. - SILAKARI, O. Synthesis and biological activity of 4-aryl-3-benzoyl-5-phenylspiro [pyrrolidine-2.3 '-indolin]-2 '-one derivatives as novel potent inhibitors of advanced glycation end product. In EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. ISSN 0223-5234; 1768-3254, 2014, vol. 79, p. 282-289. SANGSHETTI, J.N. - CHOUTHE, R.S. - SAKLE, N.S. - GONJARI, I. - SHINDE, D.B. Aldose reductase: A multi-disease target. In CURRENT ENZYME INHIBITION. ISSN 1573-4080, 2014, vol. 10, no. 1, p. 2-12 MACCARI, R. - OTTANA, R. Targeting aldose reductase for the treatment of diabetes complications and inflammatory diseases: New insights and future directions. In JOURNAL OF MEDICINAL CHEMISTRY. ISSN 0022-2623, 2015, vol. 58, no. 5, p. 2047-2067. IQBAL, Z. – HAMEED, S. – ALI, S. – TEHSEEN, Y. – SHAHID, M. – IQBAL, J. Synthesis, characterization, hypoglycemic and aldose reductase inhibition activity of arylsulfonylspiro[fluorene-9,5′-imidazolidine]-2′,4′-diones. In EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. ISSN 0223-5234, 2015, vol. 98, p. 127-138. GREWAL, A.S. - BHARDWAJ, S. - PANDITA, D. - LATHER, V. - SEKHON, B.S. Updates on aldose reductase inhibitors for management of diabetic complications and non-diabetic diseases. In MINI-REVIEWS IN MEDICINAL CHEMISTRY. ISSN 1389-5575, 2016, vol. 16, no. 2, p. 120-162. ZHU, S.J. - HAO, X. - ZHANG, S.Z. - QIN, X.Y. - CHEN, X. - ZHU, C.J. Synthesis of benzothiadiazine derivatives exhibiting dual activity as aldose reductase inhibitors and antioxidant agents. In BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. ISSN 0960-894X, 2016, vol. 26, no. 12, p. 2880-2885. GOPINATH, G. - SANKESHI, V. - PERUGU, S. - ALAPARTHI, M.D. - BANDARU, S. - PASALA, V.K. - CHITTINENI, P.R. - KRUPADANAM, G.L.D. - SAGURTHI, S.R. Design and synthesis of chiral 2H-chromene-N-imidazolo-amino acid conjugates as aldose reductase inhibitors. In EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. ISSN 0223-5234, 2016, vol. 124, p. 750-762. ZHU, S.J. - ZHANG, S.Z. - HAO, X. - QIN, X.Y. - PARVEEN, S. - YANG, S.Q. - MA, B. - ZHU, C.J. Pyridothiadiazine derivatives as aldose reductase inhibitors having antioxidant activity. In JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY. ISSN 1475-6366, 2016, vol. 31, p. 126-130. GRIBBLE, G.W. Indole ring synthesis: From natural products to drug discovery. (Book). In INDOLE RING SYNTHESIS: FROM NATURAL PRODUCTS TO DRUG DISCOVERY. Wiley, 2016, p. 1-688. ISBN 978-111869569-2;978-047051218-0 MILACKOVA, I. - KAPUSTOVA, K. - MUCAJI, P. - HOSEK, J. Artichoke leaf extract inhibits AKR1B1 and reduces NF-kappa B activity in human leukemic cells. In PHYTOTHERAPY RESEARCH. ISSN 0951-418X, 2017, vol. 31, no. 3, p. 488-496. MILACKOVA, I. - MESCANOVA, M. - SEVCIKOVA, V. - MUCAJI, P. Water leaves extracts of Cornus mas and Cornus kousa as aldose reductase inhibitors: The potential therapeutic agents. In CHEMICAL PAPERS. ISSN 0366-6352, 2017, vol. 71, no. 12, p. 2335-2341. SALEM, M.G. - AZIZ, Y.M.A. - ELEWA, M. - ELSHIHAWY, H.A. - SAID, M.M. Molecular modelling and synthesis of spiroimidazolidine-2,4-diones with dual activities as hypoglycemic agents and selective inhibitors of aldose reductase. In BIOORGANIC CHEMISTRY. ISSN 0045-2068, SEP 2018, vol. 79, p. 131-144. TASLIMI, P. - ASLAN, H.E. - DEMIR, Y. - OZTASKIN, N. - MARAS, A. - GULCIN, I. - BEYDEMIR, S. - GOKSU, S. Diarylmethanon, bromophenol and diarylmethane compounds: Discovery of potent aldose reductase, alpha-amylase and alpha-glycosidase inhibitors as new therapeutic approach in diabetes and functional hyperglycemia. In INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES. ISSN 0141-8130, NOV 2018, vol. 119, p. 857-863. IQBAL, Z. - MORAHAN, G. - AROOJ, M. - SOBOLEV, A.N. - HAMEED, S. Synthesis of new arylsulfonylspiroimidazolidine-2 ',4 '-diones and study of their effect on stimulation of insulin release from MIN6 cell line, inhibition of human aldose reductase, sorbitol accumulations in various tissues and oxidative stress. In EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. ISSN 0223-5234, 2019, vol. 168, p. 154-175. SALEM, M.G. - AZIZ, Y.M.A. - ELEWA, M. - ELSHIHAWY, H.A. - SAID, M.M. Synthesis and molecular modeling of novel non-sulfonylureas as hypoglycemic agents and selective ALR2 inhibitors. In BIOORGANIC & MEDICINAL CHEMISTRY. ISSN 0968-0896, 2019, vol. 27, no. 15, p. 3383-3389. HUANG, W.R. - ZHANG, Y. - LIANG, X. - YANG, L.C. Substituted 2-thioxothiazolidin-4-one derivatives showed protective effects against diabetic cataract via inhibition of aldose reductase. In ARCHIV DER PHARMAZIE. ISSN 0365-6233, 2020, vol. 353, no. 6, art. no. e1900371. FORMAN, V. - SUSANIKOVA, I. - KUKUROVA, L. - SVAJDLENKA, E. - NAGY, M. - MUCAJI, P. Flower Infusions From Cornus mas and Cornus kousa Inhibit Aldose Reductase Enzyme, Without Any Effects on Lipotoxicity. In NATURAL PRODUCT COMMUNICATIONS. ISSN 1934-578X, 2020, vol. 15, no. 3. VYAS, B. - CHOUDHARY, S. - SINGH, P.K. - KUMAR, M. - VERMA, H. - SINGH, M. - MALIK, A.K. - SILAKARI, O. Search for non-acidic ALR2 inhibitors: Evaluation of flavones as targeted agents for the management of diabetic complications. In BIOORGANIC CHEMISTRY. ISSN 0045-2068, 2020, vol. 96, art. no. 103570. KOUSAXIDIS, A. - PETROU, A. - LAVRENTAKI, V. - FESATIDOU, M. - NICOLAOU, I. - GERONIKAKI, A. Aldose reductase and protein tyrosine phosphatase 1B inhibitors as a promising therapeutic approach for diabetes mellitus. In EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. ISSN 0223-5234, 2020, vol. 207, art. no. 112742. SALEM, M.G. - AZIZ, Y.M.A. - ELEWA, M. - NAFIE, M.S. - ELSHIHAWY, H.A. - SAID, M.M. Synthesis, molecular modeling, selective aldose reductase inhibition and hypoglycemic activity of novel meglitinides. In BIOORGANIC CHEMISTRY. ISSN 0045-2068, 2021, vol. 111. ZHANG, Xiaonan - CHEN, Huan - ZHANG, Xin - XU, Long - LEI, Yanqi - LIU, Wenchao - LI, Lingyun - XU, Hulin - ZHU, Changjin - MA, Bing. beta-Aldehyde ketones as dual inhibitors of aldose reductase and alpha-glucosidase with antioxidant properties. In NEW JOURNAL OF CHEMISTRY. ISSN 1144-0546, 2022, vol. 46, no. 13, pp. 6165-6173. Dostupné na: https://doi.org/10.1039/d1nj03426j. AYOUP, Mohammed Salah - KHALED, Nourhan - ABDEL-HAMID, Hamida - GHAREEB, Doaa A. - NASR, Samah A. - OMER, Ahmed - SONOUSI, Amr - KASSAB, Asmaa E. - ELTAWEIL, Abdelazeem S. Novel sulfonamide derivatives as multitarget antidiabetic agents: design, synthesis, and biological evaluation. In RSC ADVANCES. FEB 29 2024, vol. 14, no. 11, p. 7664-7675. Dostupné na: https://doi.org/10.1039/d4ra01060d. Category ADCA - Scientific papers in foreign journals registered in Current Contents Connect with IF (impacted) Category of document (from 2022) V3 - Vedecký výstup publikačnej činnosti z časopisu Type of document článok Year 2008 Registered in WOS Registered in SCOPUS Registered in CCC DOI 10.1016/j.bmc.2008.03.039 
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rok CC IF IF Q (best) JCR Av Jour IF Perc SJR SJR Q (best) CiteScore A rok vydania rok metriky IF IF Q (best) SJR SJR Q (best) 2008 2007 2.662 Q2 1.062 Q1
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