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Enhancing activity and selectivity in a series of pyrrol-1-yl-1-hydroxypyrazole-based aldose reductase inhibitors: The case of trifluoroacetylation
Title Enhancing activity and selectivity in a series of pyrrol-1-yl-1-hydroxypyrazole-based aldose reductase inhibitors: The case of trifluoroacetylation Author Papastavrou Nikolaos Co-authors Chatzopoulou Maria Balleková Jana 1989- SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV SCOPUS Cappiello Mario Moschini Roberta Balestri Francesco Patsilinakos Alexandros Ragno Rino Štefek Milan 1950-2023 SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV SCOPUS ORCID Nicolaou Ioannis Source document European Journal of Medicinal Chemistry. Vol. 130 (2017), p. 328-335 Language eng - English Country FR - France Document kind rozpis článkov z periodík (rbx) Citations TASLIMI, P. - ASLAN, H.E. - DEMIR, Y. - OZTASKIN, N. - MARAŞ, A. - GULÇIN, İ. - BEYDEMIR, S. - GOKSU, S. Diarylmethanon, bromophenol and diarylmethane compounds: Discovery of potent aldose reductase, α-amylase and α-glycosidase inhibitors as new therapeutic approach in diabetes and functional hyperglycemia. In INTERNATIONAL JOURNAL OF BIOLOGICAL MACROMOLECULES. ISSN 0141-8130, 2018, vol. 119, p. 857-863. HAN, Z.F. - ZHU, J.K. - ZHANG, Y.N. - ZHANG, Y. - ZHANG, H.Y. - QI, G. - ZHU, C.J. - HAO, X. Novel quinolin-4(1H)-one derivatives as multi-effective aldose reductase inhibitors for treatment of diabetic complications: Synthesis, biological evaluation, and molecular modeling studies. In BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. ISSN 0960-894X, 2020, vol. 30, no. 9, art. no. 127101. HAN, Z.F. - QI, G. - ZHU, J.K. - ZHANG, Y.D. - XU, Y. - YAN, K. - ZHU, C.J. - HAO, X. Novel 3,4-dihydroquinolin-2(1 H )-one derivatives as dual inhibitor targeting AKR1B1/ROS for treatment of diabetic complications: Design, synthesis and biological evaluation. In BIOORGANIC CHEMISTRY. ISSN 0045-2068, 2020, vol. 105, art. no. 104428. REDDY, G.M. - CAMILO, A. - GARCIA, J.R. Pyrrole-2,5-dione analogs as a promising antioxidant agents: microwave-assisted synthesis, bio-evaluation, SAR analysis and DFT studies/interpretation. In BIOORGANIC CHEMISTRY. ISSN 0045-2068, 2021, vol. 106, art. no. 104465. MALLIKARJUNA REDDY, G. - CAMILO, A. - RAUL GARCIA, J. Pyrrole-2,5-dione analogs as a promising antioxidant agents: microwave-assisted synthesis, bio-evaluation, SAR analysis and DFT studies/interpretation. In Bioorganic Chemistry. ISSN 00452068, 2021-01-01, 106, pp. HORGAN, Conor - O'SULLIVAN, Timothy P. Recent Developments in the Practical Application of Novel Carboxylic Acid Bioisosteres. In CURRENT MEDICINAL CHEMISTRY, 2022, vol. 29, no. 13, pp. 2203-2234. ISSN 0929-8673. Dostupné na: https://doi.org/10.2174/0929867328666210820112126. YAHYA, S. - HAIDER, K. - PATHAK, A. - CHOUDHARY, A. - HOODA, P. - SHAFEEQ, M. - YAR, M.S. Strategies in synthetic design and structure-activity relationship studies of novel heterocyclic scaffolds as aldose reductase-2 inhibitors. In ARCHIV DER PHARMAZIE. ISSN 0365-6233, DEC 2022, vol. 355, no. 12. Dostupné na: https://doi.org/10.1002/ardp.202200167. HAN, Zhongfei - LI, Jiahui - XU, Zilu - SU, Yu - WANG, Yihan - ZHUO, Lili - DU, Jiaming - ZHU, Changjin - HAO, Xin. Design and synthesis of novel quinazolin-4(1H)-one derivatives as potent and selective inhibitors targeting AKR1B1. In Archiv der Pharmazie, 2023-04-01, 356, 4, pp. ISSN 03656233. Dostupné na: https://doi.org/10.1002/ardp.202200577. Category ADCA - Scientific papers in foreign journals registered in Current Contents Connect with IF (impacted) Category of document (from 2022) V3 - Vedecký výstup publikačnej činnosti z časopisu Type of document článok Year 2017 Registered in WOS Registered in SCOPUS Registered in CCC DOI 10.1016/j.ejmech.2017.02.053 
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File name Access Size Downloaded Type License Enhancing activity and selectivity in a series of pyrrol-1-yl-1-hydroxypyrazole-based aldose reductase inhibitors The case of trifluoroacetylation.pdf Neprístupný/archív 1.3 MB 1 Publisher's version rok CC IF IF Q (best) JCR Av Jour IF Perc SJR SJR Q (best) CiteScore A rok vydania rok metriky IF IF Q (best) SJR SJR Q (best) 2017 2016 4.519 Q1 1.289 Q1
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