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Development of Novel Oxotriazinoindole Inhibitors of Aldose Reductase: Isosteric Sulfur/Oxygen Replacement in the Thioxotriazinoindole Cemtirestat Markedly Improved Inhibition Selectivity
Title Development of Novel Oxotriazinoindole Inhibitors of Aldose Reductase: Isosteric Sulfur/Oxygen Replacement in the Thioxotriazinoindole Cemtirestat Markedly Improved Inhibition Selectivity Author Hlaváč Matúš 1991- Co-authors Kováčiková Lucia 1983- SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV SCOPUS ORCID Šoltésová Prnová Marta 1986- SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV SCOPUS ORCID Šramel Peter 1989- Addová Gabriela 1974- Májeková Magdaléna 1958- SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV SCOPUS RID ORCID Hanquet Gilles Boháč Andrej 1964- Štefek Milan 1950-2023 SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV SCOPUS ORCID Source document Journal of Medicinal Chemistry. Vol. 63, no. 1 (2020), p. 369-381 Language eng - English Country US - United States of America Note APVV SK-FR-2015-0014, TUBITAK project no: 215S19, Vega 1/0670/18 Document kind rozpis článkov z periodík (rbx) Citations VALACHOVA, K. - MACH, M. - SOLTES, L. Oxidative Degradation of High-Molar-Mass Hyaluronan: Effects of Some Indole Derivatives to Hyaluronan Decay. In INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES. eISSN: 1422-0067, 2020, vol. 21, no. 16, art. no. 5609. CHEN, Q.F. - PAN, Y.H. - YUE, T.T. - YANG, W.R. - LIU, H. - ZHENG, J. [4+2]-Annulation of Prop-2-ynylsulfonium Salts and Isatoic Anhydrides: Access to 3-Methylthio-4-quinolones. In ORGANIC LETTERS. ISSN 1523-7060, 2020, vol. 22, no. 15, p. 6096-6100. HAN, Z.F. - QI, G. - ZHU, J.K. - ZHANG, Y.D. - XU, Y. - YAN, K. - ZHU, C.J. - HAO, X. Novel 3,4-dihydroquinolin-2(1 H )-one derivatives as dual inhibitor targeting AKR1B1/ROS for treatment of diabetic complications: Design, synthesis and biological evaluation. In BIOORGANIC CHEMISTRY. ISSN 0045-2068, 2020, vol. 105, art. no. 104428. KOUSAXIDIS, A. - PETROU, A. - LAVRENTAKI, V. - FESATIDOU, M. - NICOLAOU, I. - GERONIKAKI, A. Aldose reductase and protein tyrosine phosphatase 1B inhibitors as a promising therapeutic approach for diabetes mellitus. In EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. ISSN 0223-5234, 2020, vol. 207, art. no. 112742. CHEN, H. - ZHANG, X. - ZHANG, X.N. - LIU, W.C. - LEI, Y.Q. - ZHU, C.J. - MA, B. (5-Hydroxy-4-oxo-2-styryl-4H-pyridin-1-yl)-acetic Acid Derivatives as Multifunctional Aldose Reductase Inhibitors. In MOLECULES. eISSN: 1420-3049, 2020, vol. 25, no. 21, art. no. 5135. IMRAN, Aqeel - SHEHZAD, Muhammad Tariq - AL ADHAMI, Taha - RAHMAN, Khondaker Miraz - HUSSAIN, Dilawar - ALHARTHY, Rima D. - SHAFIQ, Zahid - IQBAL, Jamshed. Development of coumarin-thiosemicarbazone hybrids as aldose reductase inhibitors: Biological assays, molecular docking, simulation studies and ADME evaluation. In BIOORGANIC CHEMISTRY. ISSN 0045-2068, 2021, vol. 115, no., pp. Dostupné na: https://doi.org/10.1016/j.bioorg.2021.105164. HIEBEL, Marie Aude - SUZENET, Franck. Triazines, tetrazines, and fused ring polyaza systems. In Progress in Heterocyclic Chemistry. ISSN 09596380, 2021-01-01, 33, pp. 441-472. Dostupné na: https://doi.org/10.1016/B978-0-323-98410-2.00014-X. LU, Nan - LIANG, Hui - MIAO, Chengxia - LAN, Xiaozheng - QIAN, Ping. Theoretical investigation of the mechanism of DMAP-promoted [4+2]-annulation of prop-2-ynylsulfonium with isatoic anhydride. In CANADIAN JOURNAL OF CHEMISTRY. ISSN 0008-4042, 2022, vol. 100, no. 4, pp. 263-271. Dostupné na: https://doi.org/10.1139/cjc-2021-0174. KUMAR, Hariom - DHAMEJA, Manoj - KURELLA, Sirisha - UMA, Adepally - GUPTA, Preeti. Synthesis, in-vitro alpha-glucosidase inhibition and molecular docking studies of 1,3,4-thiadiazole-5,6-diphenyl-1,2,4-triazine hybrids: Potential leads in the search of new antidiabetic drugs. In JOURNAL OF MOLECULAR STRUCTURE, 2023, vol. 1273, no., pp. ISSN 0022-2860. Dostupné na: https://doi.org/10.1016/j.molstruc.2022.134339. HAN, Zhongfei - LI, Jiahui - XU, Zilu - SU, Yu - WANG, Yihan - ZHUO, Lili - DU, Jiaming - ZHU, Changjin - HAO, Xin. Design and synthesis of novel quinazolin-4(1H)-one derivatives as potent and selective inhibitors targeting AKR1B1. In ARCHIV DER PHARMAZIE, 2023, vol. 356, no. 4, pp. ISSN 0365-6233. Dostupné na: https://doi.org/10.1002/ardp.202200577. ZHAO, W.H. - XU, J.H. - TANGADANCHU, V.K.R. - ZHOU, C.H. Thiazolyl hydrazineylidenyl indolones as unique potential multitargeting broad-spectrum antimicrobial agents. In EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. ISSN 0223-5234, AUG 5 2023, vol. 256. Dostupné na: https://doi.org/10.1016/j.ejmech.2023.115452. Category ADCA - Scientific papers in foreign journals registered in Current Contents Connect with IF (impacted) Category of document (from 2022) V3 - Vedecký výstup publikačnej činnosti z časopisu Type of document článok Year 2020 Registered in WOS Registered in SCOPUS Registered in CCC DOI 10.1021/acs.jmedchem.9b01747 
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File name Access Size Downloaded Type License Development of Novel Oxotriazinoindole Inhibitors of Aldose Reductase Isosteric Sulfur.pdf Neprístupný/archív 1.6 MB 1 Publisher's version rok CC IF IF Q (best) JCR Av Jour IF Perc SJR SJR Q (best) CiteScore A rok vydania rok metriky IF IF Q (best) SJR SJR Q (best) 2020 2019 6.205 Q1 2.093 Q1
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