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Identification of small molecule regulators of the nuclear receptor HNF4 alpha based on naphthofuran scaffolds
Title Identification of small molecule regulators of the nuclear receptor HNF4 alpha based on naphthofuran scaffolds Author Guével Rémy Le Dudášová Zuzana 1979- SAVEXONK - Ústav experimentálnej onkológie SAV Baráth Peter 1972- SAVEXONK - Ústav experimentálnej onkológie SAV SCOPUS RID ORCID Co-authors Oger Frédérik Lecorgne Aurélien Chevance Soizic Bondon Arnaud Simonneaux Gérard Salbert Gilles Source document Bioorganic & Medicinal Chemistry. Vol. 17, no. 19 (2009), p. 7021-7030 Language eng - English Country US - United States of America Document kind rozpis článkov z periodík (rbx) Citations TSAI, Yi-Ling - DAS, Utpal - SYU, Siang-en - LEE, Chia-Jui - LIN, Wenwei. Facile Synthesis of Functional Tricyclic Fused Furans by Intramolecular Wittig Reactions. In EUROPEAN JOURNAL OF ORGANIC CHEMISTRY. ISSN 1434-193X, 2013, vol. 2013, no. 21, pp. 4634. XIA, Likai - MAGAR, Krishna Bahadur Somai - LEE, Yong Rok. Synthesis of novel and diverse naphtho[1,2-b]furans by phosphine-catalyzed [3+2] annulation of activated 1,4-naphthoquinones and acetylenecarboxylates. In MOLECULAR DIVERSITY. ISSN 1381-1991, 2015, vol. 19, no. 1, pp. 55. CHAMOUTON, Julie - LATRUFFE, Norbert. PPAR alpha/HNF4 alpha Interplay on Diversified Responsive Elements. Relevance in the Regulation of Liver Peroxisomal Fatty Acid Catabolism. In CURRENT DRUG METABOLISM. ISSN 1389-2002, 2012, vol. 13, no. 10, pp. 1436. RAO, V. Kameshwara - SHELKE, Ganesh M. - TIWARI, Rakesh - PARANG, Keykavous - KUMAR, Anil. A Simple and Efficient Synthesis of 2,3-Diarylnaphthofurans Using Sequential Hydroarylation/Heck Oxyarylation. In ORGANIC LETTERS. ISSN 1523-7060, 2013, vol. 15, no. 9, pp. 2190. CHENG, Bao - LIN, Yongsheng - KUANG, Ming - FANG, Sai - GU, Qiong - XU, Jun - WANG, Laiyou. Synthesis and Anti-neuroinflammatory Activity of Lactone Benzoyl Hydrazine and 2-nitro-1-phenyl-1 H-Indole Derivatives as p38 alpha MAPK Inhibitors. 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KISELYUK, Alice - LEE, Seung-Hee - FARBER-KATZ, Suzette - ZHANG, Mingjun - ATHAVANKAR, Sonalee - COHEN, Tom - PINKERTON, Anthony B. - YE, Mao - BUSHWAY, Paul - RICHARDSON, Adam D. - HOSTETLER, Heather A. - RODRIGUEZ-LEE, Mariam - HUANG, Li - SPANGLER, Benjamin - SMITH, Layton - HIGGINBOTHAM, Jennifer - CASHMAN, John - FREEZE, Hudson - ITKIN-ANSARI, Pamela - DAWSON, Marcia I. - SCHROEDER, Friedhelm - CANG, Yong - MERCOLA, Mark - LEVINE, Fred. HNF4 alpha Antagonists Discovered by a High-Throughput Screen for Modulators of the Human Insulin Promoter. In CHEMISTRY & BIOLOGY. ISSN 1074-5521, 2012, vol. 19, no. 7, pp. 806. KOEHLER, Angela N. A complex task? Direct modulation of transcription factors with small molecules. In CURRENT OPINION IN CHEMICAL BIOLOGY. ISSN 1367-5931, 2010, vol. 14, no. 3, pp. 331. 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Design and synthesis of 2,3-dihydro- and 5-chloro-2,3-dihydro-naphtho-[1,2-b]furan-2-carboxylic acid N-(substitutedphenyl)amide analogs and their biological activities as inhibitors of NF-kappa B activity and anticancer agents. In ARCHIVES OF PHARMACAL RESEARCH. ISSN 0253-6269, MAY 2016, vol. 39, no. 5, p. 618-630. KWON, S.M. - JUNG, Y.Y. - HWANG, C.J. - PARK, M.H. - YOON, N.Y. - KIM, T.M. - YU, J.M. - KIM, D.H. - SEO, D.W. - YOUN, H.S. - SEO, H.O. - CHUNG, I.S. - HAN, S.B. - HWANG, B.Y. - YOO, H.S. - JUNG, J.K. - LEE, H. - HONG, J.T. Anti-cancer effect of N-(3,5-bis(trifluoromethyl)phenyl)-5-chloro-2,3-dihydronaphtho[1,2-b]fur an-2-carboxamide, a novel synthetic compound. In MOLECULAR CARCINOGENESIS. ISSN 0899-1987, MAY 2016, vol. 55, no. 5, p. 659-670. HUANG, Jin - WANG, Wei - HE, Hai-Yu - JIAN, Lei - FU, Hai-Yan - ZHENG, Xue-Li - CHEN, Hua - LI, Rui-Xiang. An Approach to the Synthesis of 1-Propenylnaphthols and 3-Arylnaphtho[2,1-b]furans. In JOURNAL OF ORGANIC CHEMISTRY. 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Cascade Rh(ii) and Yb(iii) catalyzed synthesis of substituted naphthofurans via transannulation of N-sulfonyl-1,2,3-triazoles with beta-naphthols. In CHEMICAL COMMUNICATIONS. ISSN 1359-7345, 2019, vol. 55, no. 31, pp. 4507-4510. JAYARAJAN, Ramasamy - KUMAR, Rakesh - GUPTA, Jagriti - DEV, Gayathri - KADU, Pradeep - CHATTERJEE, Debdeep - BAHADUR, Dhirendra - MAITI, Debabrata - MAJI, Samir K. Fabrication of an amyloid fibril-palladium nanocomposite: a sustainable catalyst for C-H activation and the electrooxidation of ethanol. In JOURNAL OF MATERIALS CHEMISTRY A. ISSN 2050-7488, 2019, vol. 7, no. 9, pp. 4486-4493. TAKAHASHI, Shuhei - SHIMOOKA, Hirokazu - OKAUCHI, Tatsuo - KITAMURA, Mitsuru. Pd-catalyzed Cyclization of Terminal Alkynes using Diazonaphthoquinones: Synthesis of Naphtho[1,2-b]furans. In CHEMISTRY LETTERS. ISSN 0366-7022, 2019, vol. 48, no. 1, pp. 28-31. SINGH, Puja - TUNG, Shu-Ping - HAN, Eun Hee - LEE, In-Kyu - CHI, Young-In. 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Domino Reaction of 2,4-Diyn-1-ols with 1,3-Dicarbonyl Compounds: Direct Access to Aryl/Heteroaryl-Fused Benzofurans and Indoles. In ORGANIC LETTERS. ISSN 1523-7060, JUN 18 2021, vol. 23, no. 12, p. 4882-4887. RAJESH, P. - ALMANSOUR, A.I. - ARUMUGAM, N. - YARAGORLA, S. Calcium-catalyzed formal [3+2] annulation of C,N-diacyliminium ions with nucleophilic phenols: a diversity oriented synthesis of 3-aminofurans. In ORGANIC & BIOMOLECULAR CHEMISTRY. ISSN 1477-0520, FEB 7 2021, vol. 19, no. 5, p. 1060-1065. BENZI, A. - BIANCHI, L. - GIORGI, G. - MACCAGNO, M. - PETRILLO, G. - SPINELLI, D. - TAVANI, C. An Easy Access to Furan-Fused Polyheterocyclic Systems. In MOLECULES. MAY 2022, vol. 27, no. 10. Dostupné na: https://doi.org/10.3390/molecules27103147. GAYYUR - CHOUDHARY, S. - KANT, R. - GHOSH, N. Synergetic copper/zinc catalysis: synthesis of aryl/heteroaryl-fused 1H-pyrrolo[3,2-c]pyridines. In CHEMICAL COMMUNICATIONS. ISSN 1359-7345, FEB 8 2022, vol. 58, no. 12, p. 1974-1977. Dostupné na: https://doi.org/10.1039/d1cc05514c. LEE, S.H. - VEERIAH, V. - LEVINE, F. A potent HNF4 alpha agonist reveals that HNF4 alpha controls genes important in inflammatory bowel disease and Paneth cells. In PLOS ONE. ISSN 1932-6203, 2022, vol. 17, no. 4. Dostupné na: https://doi.org/10.1371/journal.pone.0266066. Category ADCA - Scientific papers in foreign journals registered in Current Contents Connect with IF (impacted) Category of document (from 2022) V3 - Vedecký výstup publikačnej činnosti z časopisu Type of document článok Year 2009 Registered in WOS DOI 10.1016/j.bmc.2009.07.079 
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rok CC IF IF Q (best) JCR Av Jour IF Perc SJR SJR Q (best) CiteScore A rok vydania rok metriky IF IF Q (best) SJR SJR Q (best) 2009 2008 3.075 Q1 1.206 Q1
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