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Structure-activity relations on [1-(3,5-difluoro-4-hydroxyphenyl)-1H-pyrrol-3-yl]phenylmethanone. The effect of methoxy substitution on aldose reductase inhibitory activity and selectivity
Title Structure-activity relations on [1-(3,5-difluoro-4-hydroxyphenyl)-1H-pyrrol-3-yl]phenylmethanone. The effect of methoxy substitution on aldose reductase inhibitory activity and selectivity Author Chatzopoulou Maria Co-authors Mamadou Eduard Jusková Mária 1983- SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV SCOPUS SCOPUS Koukoulitsa Cathrine Nicolaou Ioannis Štefek Milan 1950-2023 SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV SCOPUS ORCID Demopoulos Vassilis J. Source document Bioorganic & Medicinal Chemistry. Vol. 19, no. 4 (2011), p. 1426-1433 Language eng - English Country GB - Great Britian Document kind rozpis článkov z periodík (rbx) Citations ZANATTA, N. - AQUINO, E.D. - DA SILVA, F.M. - BONACORSO, H.G. - MARTINS, M.A.P. Improved One-Pot Synthesis of 1-Aryl-3-trifluoroacetyl-1H-pyrroles under Swern Oxidation. In SYNTHESIS-STUTTGART. ISSN 0039-7881, 2012, vol. 44, no. 22, p. 3477-3482. ALI, S. - SAEED, A. - ABBAS, N. - SHAHID, M. - BOLTE, M. - IQBAL, J. Design, synthesis and molecular modelling of novel methyl[4-oxo-2-(aroylimino)-3-(substituted phenyl)thiazolidin-5-ylidene]acetates as potent and selective aldose reductase inhibitors. In MEDCHEMCOMM. ISSN 2040-2503, 2012, vol. 3, no. 11, p. 1428-1434. IQBAL, Z. - ALI, S. - IQBAL, J. - ABBAS, Q. - QURESHI, I.Z. - HAMEED, S. Dual action spirobicycloimidazolidine-2,4-diones: Antidiabetic agents and inhibitors of aldose reductase-an enzyme involved in diabetic complications. In BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. ISSN 0960-894X, 2013, vol. 23, no. 2, p. 488-491. POSTIKOVA, S. - SABBAH, M. - WIGHTMAN, D. - NGUYEN, I.T. - SANSELME, M. - BESSON, T. - BRIERE, J.F. - OUDEYER, S. - LEVACHER, V. Developments in Meyers' Lactamization Methodology: En Route to Bi(hetero)aryl Structures with Defined Axial Chirality. In JOURNAL OF ORGANIC CHEMISTRY. ISSN 0022-3263, 2013, vol. 78, no. 16, p. 8191-8197. REDDY, T. N. - RAVINDER, M. - BAGUL, P. - RAVIKANTI, K. - BAGUL, Ch. - NANUBOLU, J. B. - SRINIVAS, K. - BANERJEE, S. K. - RAO, V. J. Synthesis and biological evaluation of new epalrestat analogues as aldose reductase inhibitors (ARIs). In EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. ISSN 0223-5234; 1768-3254, 2014, vol. 71, p. 53-66. OVAIS, S. - PUSHPALATHA, H. - REDDY, G. B. - RATHORE, P. - BASHIR, R. - YASEEN, S. - DHEYAA, A. - YASEEN, R. - TANWAR, O. - AKTHAR, M. - SAMIM, M. - JAVED, K. Synthesis and biological evaluation of some new pyrazoline substituted benzenesulfonylurea/thiourea derivatives as anti-hyperglycaemic agents and aldose reductase inhibitors. In EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. ISSN 0223-5234; 1768-3254, 2014, vol. 80, p. 209-217. MACCARI, R. - OTTANA, R. Targeting aldose reductase for the treatment of diabetes complications and inflammatory diseases: New insights and future directions. In JOURNAL OF MEDICINAL CHEMISTRY. ISSN 0022-2623, 2015, vol. 58, no. 5, p. 2047-2067. ZOU, Y. - QIN, X.Y. - HAO, X. - ZHANG, W. - YANG, S.Q. - YANG, Y.C. - HAN, Z.F. - MA, B. - ZHU, C.J. Phenolic 4-hydroxy and 3,5-dihydroxy derivatives of 3-phenoxyquinoxalin-2(1H)-one as potent aldose reductase inhibitors with antioxidant activity. In BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS. ISSN 0960-894X, 2015, vol. 25, no. 18, p. 3924-3927. PLIOUKAS, M. - GABRIELI, C. - LAZARI, D. - KOKKALOU, E. Phytochemical analysis with the antioxidant and aldose reductase inhibitory capacities of Tephrosia humilis aerial parts' extracts. In NATURAL PRODUCT RESEARCH. ISSN 1478-6419, 2016, vol. 30, no. 12, p. 1366-1372. SUNKE, R. - NALLAPATI, S.B. - KUMAR, J.S. - KUMAR, K.S. - PAL, M. Use of AlCl3 in Friedel Crafts arylation type reactions and beyond: an overview on the development of unique methodologies leading to N-heteroarenes. In ORGANIC & BIOMOLECULAR CHEMISTRY. ISSN 1477-0520, 2017, vol. 15, no. 19, p. 4042-4057. ZHAN, J.-Y. - MA, K. - ZHENG, Q.-C. - YANG, G.-H. - ZHANG, H.-X. Exploring the interactional details between aldose reductase (AKR1B1) and 3-Mercapto-5H-1,2,4-triazino[5,6-b]indole-5-acetic acid through molecular dynamics simulations. In JOURNAL OF BIOMOLECULAR STRUCTURE & DYNAMICS. ISSN 0739-1102, 2019, vol. 37, no. 7, p. 1724-1735. HAO, Xin - QI, Gang - MA, Hongxing - ZHU, Changjin - HAN, Zhongfei. Novel 2-phenoxypyrido[3,2-b]pyrazin-3(4H)-one derivatives as potent and selective aldose reductase inhibitors with antioxidant activity. In JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY. ISSN 1475-6366, 2019, vol. 34, no. 1, pp. 1368-1372. HAO, X. - QIN, X.Y. - ZHANG, X. - MA, B. - QI, G. - YU, T.M. - HAN, Z.F. - ZHU, C.J. Identification of quinoxalin-2(1H)-one derivatives as a novel class of multifunctional aldose reductase inhibitors. In FUTURE MEDICINAL CHEMISTRY. ISSN 1756-8919, DEC 2019, vol. 11, no. 23, p. 2989-3004. MOUSSOUNI, S. - KARAKOUSI, C.V. - TSATALAS, P. - LAZARI, D. - KOKKALOU, E. Biological Studies with Phytochemical Analysis Of Cornus mas Unripe Fruits. In CHEMISTRY OF NATURAL COMPOUNDS. ISSN 0009-3130, 2020, vol. 56, no. 1. KUMAR, M. - CHOUDHARY, S. - SINGH, P.K. - SILAKARI, O. Addressing selectivity issues of aldose reductase 2 inhibitors for the management of diabetic complications. In FUTURE MEDICINAL CHEMISTRY. ISSN 1756-8919, 2020, vol. 12, no. 14, p. 1327-1358. Category ADCA - Scientific papers in foreign journals registered in Current Contents Connect with IF (impacted) Category of document (from 2022) V3 - Vedecký výstup publikačnej činnosti z časopisu Type of document článok Year 2011 Registered in WOS Registered in SCOPUS Registered in CCC DOI 10.1016/j.bmc.2011.01.009 article
rok CC IF IF Q (best) JCR Av Jour IF Perc SJR SJR Q (best) CiteScore A rok vydania rok metriky IF IF Q (best) SJR SJR Q (best) 2011 2010 2.978 Q2 1.083 Q1
Number of the records: 1