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Title Enhancing activity and selectivity in a series of pyrrol-1-yl-1-hydroxypyrazole-based aldose reductase inhibitors: The case of trifluoroacetylation Author Papastavrou Nikolaos Co-authors Chatzopoulou Maria Balleková Jana 1989- SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV Cappiello Mario Moschini Roberta Balestri Francesco Patsilinakos Alexandros Ragno Rino Štefek Milan 1950-2023 SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV Nicolaou Ioannis Action VEGA č. 2/0041/15. Deriváty kyseliny 1-indoloctovej ako inhibítory aldózareduktázy: dizajn, syntéza a biologická aktivita : 01.01.2015 - 31.12.2017 Source document European Journal of Medicinal Chemistry. Vol. 130 (2017), p. 328-335 Category ADCA - Scientific papers in foreign journals registered in Current Contents Connect with IF (impacted) Category of document (from 2022) V3 - Vedecký výstup publikačnej činnosti z časopisu Type of document článok Year 2017 DOI 10.1016/j.ejmech.2017.02.053 File name Access Size Downloaded Type License Enhancing activity and selectivity in a series of pyrrol-1-yl-1-hydroxypyrazole-based aldose reductase inhibitors The case of trifluoroacetylation.pdf Neprístupný/archív 1.3 MB 1 Publisher's version 
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Title Pyrrol-1-yl-hydroxypyrazole: a privileged scaffold for ALR2 inhibition Author Papastavrou Nikolaos Co-authors Chatzopoulou Maria Balleková Jana 1989- SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV Štefek Milan 1950-2023 SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV Nicolaou Ioannis Source document IXth Joint Meeting in Medicinal Chemistry. Abstracts : Austria - Croatia - Czech Republic - Greece - Hungary - Italy - Poland - Slovakia - Slovenia. 7-10 June 2015. Athens, Greece. non pag. P41. - Athens : Hellenic Society of Medicinal Chemistry, 2015 ; Joint Meeting in Medicinal Chemistry Category AFG - Abstracts of papers from foreign conferences Year 2015 article
Title Decreasing acidity in a series of aldose reductase inhibitors: 2-Fluoro-4-(1H-pyrrol-1-yl)phenol as a scaffold for improved membrane permeation Author Chatzopoulou Maria Co-authors Patsilinakos Alexandros Vallianatou Theodosia Šoltésová Prnová Marta 1986- SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV Žakelj Simon Ragno Rino Štefek Milan 1950-2023 SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV Kristl Albin Tsantili-Kakoulidou Anna Demopoulos Vassilis J. Action VEGA č. 2/0067/11. Molekulové modelovanie, syntéza a biologická aktivita substituovaných pyridoindolov ako bifunkčných agens v prevencii diabetických komplikácií : 2011 - 2014 Source document Bioorganic & Medicinal Chemistry. Vol. 22 (2014), p. 2194-2207 Category ADCA - Scientific papers in foreign journals registered in Current Contents Connect with IF (impacted) Category of document (from 2022) V3 - Vedecký výstup publikačnej činnosti z časopisu Type of document článok Year 2014 DOI 10.1016/j.bmc.2014.02.016 File name Access Size Downloaded Type License Decreasing acidity in a series of aldose reductase inhibitors....pdf Neprístupný/archív 2.1 MB 1 Publisher's version article
Title Structure-activity relations on [1-(3,5-difluoro-4-hydroxyphenyl)-1H-pyrrol-3-yl]phenylmethanone. The effect of methoxy substitution on aldose reductase inhibitory activity and selectivity Author Chatzopoulou Maria Co-authors Mamadou Eduard Jusková Mária 1983- SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV Koukoulitsa Cathrine Nicolaou Ioannis Štefek Milan 1950-2023 SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV Demopoulos Vassilis J. Action COST Action B35. Lipid Peroxidation Associated Disorders: LPO : 02.06.2006 - 01.06.2010 VEGA č. 2/0001/08. Substituované pyridoindoly ako inhibítory aldózareduktázy s antioxidačnou aktivitou v liečbe diabetických komplikácií: predklinické štúdium v bunkových systémoch in vitro a na diabetických potkanoch in vivo : 2008 - 2010 Source document Bioorganic & Medicinal Chemistry. Vol. 19, no. 4 (2011), p. 1426-1433 Category ADCA - Scientific papers in foreign journals registered in Current Contents Connect with IF (impacted) Category of document (from 2022) V3 - Vedecký výstup publikačnej činnosti z časopisu Type of document článok Year 2011 DOI 10.1016/j.bmc.2011.01.009 article