Počet záznamov: 1  

Cancer-Related Carbonic Anhydrase Isozymes and Their Inhibition

  1. NázovCancer-Related Carbonic Anhydrase Isozymes and Their Inhibition
    Autor Pastoreková Silvia 1961 SAVVIR - Virologický ústav SAV    ORCID
    Spoluautori Pastorek Jaromír 1957- SAVVIR - Virologický ústav SAV

    Zdroj.dok. Carbonic Anhydrase. Its Inhibitors and Activators : CRC Enzyme Inhibitors Series. P. 255 - 281. - Boca Raton, Florida : CRC Press, 2004 / Supuran C.T. ; Scozzafava A. ; Conway J.
    Jazyk dok.eng - angličtina
    KrajinaUS - Spojené štáty
    Druh dok.rozpis článkov z periodík (rzb)
    OhlasyScozzafava, A; Mastrolorenzo, A; Supuran, CT Modulation of carbonic anhydrase activity and its applications in therapy Modulation of carbonic anhydrase activity and its applications in therapy EXPERT OPINION ON THERAPEUTIC PATENTS Volume: 14 Issue: 5 Pages: 667-702 Published: MAY 2004
    Garaj, V (Garaj, V); Puccetti, L (Puccetti, L); Fasolis, G (Fasolis, G); Winum, JY (Winum, JY); Montero, JL (Montero, JL); Scozzafava, A (Scozzafava, A); Vullo, D (Vullo, D); Innocenti, A (Innocenti, A); Supuran, CT (Supuran, CT) Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides incorporating 1,2,4-triazine moieties BIOORGANIC & MEDICINAL CHEMISTRY LETTERS Volume: 14 Issue: 21 Pages: 5427-5433, 2004
    Winum, JY (Winum, JY); Dogne, JM (Dogne, JM); Casini, A (Casini, A); de Leval, X (de Leval, X); Montero, JL (Montero, JL); Scozzafava, A (Scozzafava, A); Vullo, D (Vullo, D); Innocenti, A (Innocenti, A); Supuran, CT (Supuran, CT) Carbonic anhydrase inhibitors: Synthesis and inhibition of cytosolic membrane-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides incorporating hydrazino moieties JOURNAL OF MEDICINAL CHEMISTRY Volume: 48 Issue: 6 Pages: 2121-2125, 2005
    Vullo, D (Vullo, D); Steffansen, B (Steffansen, B); Brodin, B (Brodin, B); Supuran, CT (Supuran, CT); Scozzafava, A (Scozzafava, A); Nielsen, CU Carbonic anhydrase inhibitors: Transepithelial transport of thioureido sulfonamide inhibitors of the cancer-associated isozyme IX is dependent on efflux transporters BIOORGANIC & MEDICINAL CHEMISTRY Volume: 14 Issue: 7 Pages: 2418-2427, 2006
    Thiry, A (Thiry, A); Ledecq, M (Ledecq, M); Cecchi, A (Cecchi, A); Dogne, JM (Dogne, JM); Wouters, J (Wouters, J); Supuran, CT (Supuran, CT); Masereel, B Indanesulfonamides as carbonic anhydrase inhibitors. Toward structure-based design of selective inhibitors of the tumor-associated isozyme CA IX JOURNAL OF MEDICINAL CHEMISTRY Volume: 49 Issue: 9 Pages: 2743-2749, 2006
    Zareef, M (Zareef, Muhammad); Innocenti, A (Innocenti, Alessio); Iqbal, R (Iqbal, Rashid); Zaidi, JH (Zaidi, Javid H.); Arfan, M (Arfan, Muhammad); Scozzafava, A (Scozzafava, Andrea); Supuran, CT (Supuran, Claudiu T.) Carbonic anhydrase inhibitors. Inhibition of human tumor-associated isozymes IX and cytosolic isozymes I and II with some 1,3,4-oxadiazole-thiols JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY Volume: 21 Issue: 4 Pages: 351-359, 2006
    Saczewski, F (Saczewski, Franciszek); Innocenti, A (Innocenti, Alessio); Brzozowski, Z (Brzozowski, Zdzislaw); Slawinski, J (Slawinski, Jaroslaw); Pomarnacka, E (Pomarnacka, Elzbieta); Kornicka, A (Kornicka, Anita); Scozzafava, A (Scozzafava, Andrea); Supuran, CT (Supuran, Claudiu T.) Carbonic anhydrase inhibitors. Selective inhibition of human tumor-associated isozymes IX and XII and cytosolic isozymes I and II with some substituted-2-mercapto-benzenesulfonamides JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY Volume: 21 Issue: 5 Pages: 563-568, 2006
    Thiry, A (Thiry, Anne); Dogne, JM (Dogne, Jean-Michel); Masereel, B (Masereel, Bernard); Supuran, CT (Supuran, Claudiu T.) Targeting tumor-associated carbonic anhydrase IX in cancer therapy TRENDS IN PHARMACOLOGICAL SCIENCES Volume: 27 Issue: 11 Pages: 566-573, 2006
    Ozensoy, Ozen; Supuran, Claudiu T. arbonic anhydrase IX as prognostic marker for tumor progression and as a target for novel antitumor drugs TURKISH JOURNAL OF BIOCHEMISTRY-TURK BIYOKIMYA DERGISI Volume: 32 Issue: 3 Pages: 130-134 Published: 2007
    Dogne, JM (Dogne, Jean-Michel); Thiry, A (Thiry, Anne); Pratico, D (Pratico, Domenico); Masereel, B (Masereel, Bernard); Supuran, CT Dual carbonic anhydrase - Cyclooxygenase-2 inhibitors CURRENT TOPICS IN MEDICINAL CHEMISTRY Volume: 7 Issue: 9 Pages: 885-891, 2007
    Thiry, A (Thiry, Anne); Dogne, J (Dogne, Jean-Michel); Supuran, CT (Supuran, Claudiu T.); Masereel, B (Masereel, Bernard) Carbonic anhydrase inhibitors as anticonvulsant agents CURRENT TOPICS IN MEDICINAL CHEMISTRY Volume: 7 Issue: 9 Pages: 855-864, 2007
    Nuti, E (Nuti, Elisa); Orlandini, E (Orlandini, Elisabetta); Nencetti, S (Nencetti, Susanna); Rossello, A (Rossello, Armando); Innocenti, A (Innocenti, Alessio); Scozzafava, A (Scozzafava, Andrea); Supuran, CT (Supuran, Claudiu T.) Carbonic anhydrase and matrix metalloproteinase inhibitors. Inhibition of human tumor-associated isozymes IX and cytosolic isozyme I and II with sulfonylated hydroxamates IOORGANIC & MEDICINAL CHEMISTRY Volume: 15 Issue: 6 Pages: 2298-2311, 2007
    Colinas, PA (Colinas, Pedro A.); Bravo, RD (Bravo, Rodolfo D.); Vullo, D (Vullo, Daniela); Scozzafava, A (Scozzafava, Andrea); Supuran, CT (Supuran, Claudiu T.) Carbonic anhydrase inhibitors. Inhibition of cytosolic isoforms I and II, and extracellular isoforms IV, IX, and XII with sulfamides incorporating sugar moieties BIOORGANIC & MEDICINAL CHEMISTRY LETTERS Volume: 17 Issue: 18 Pages: 5086-5090, 2007
    Anai, S (Anai, Satoshi); Shiverick, K (Shiverick, Kathleen); Medrano, T (Medrano, Theresa); Nakamura, K (Nakamura, Kogenta); Goodison, S (Goodison, Steve); Brown, BD (Brown, Bob D.); Rosser, CJ (Rosser, Charles J.) Downregulation of BCL-2 induces downregulation of carbonic anhydrase IX, vascular endothelial growth factor, and pAkt and induces radiation sensitization UROLOGY Volume: 70 Issue: 4 Pages: 832-837, 2007
    Supuran, Claudiu T. The tumor-associated metalloenzyme carbonic anhydrase IX (CA IX) as a drug target METAL IONS IN BIOLOGY AND MEDICINE, VOL 10 Book Series: METAL IONS IN BIOLOGY AND MEDICINE Volume: 10 Pages: 379-381 Published: 2008
    Ozensoy, O (Ozensoy, Ozen)[ 1 ] ; Arslan, O (Arslan, Oktay)[ 1 ] ; Kockar, F Differential in vitro inhibition effects of some antibiotics on tumor associated carbonic anhydrase isozymes of hCA-IX and hCA-XII JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY Volume: 23 Issue: 4 Pages: 579-585, 2008
    Rami, M (Rami, Marouan)[ 2 ] ; Winum, JY (Winum, Jean-Yves)[ 2 ] ; Innocenti, A (Innocenti, Alessio)[ 1 ] ; Montero, JL (Montero, Jean-Louis)[ 2 ] ; Scozzafava, A (Scozzafava, Andrea)[ 1 ] ; Supuran, CT (Supuran, Claudlu T.)[ 1 ] Carbonic anhydrase inhibitors: Copper(II) complexes of polyamino-polycarboxylamido aromatic/heterocyclic sulfonamides are very potent inhibitors of the tumor-associated isoforms IX and XII BIOORGANIC & MEDICINAL CHEMISTRY LETTERS Volume: 18 Issue: 2 Pages: 836-841, 2008
    Supuran, Claudiu T. Carbonic anhydrases: novel therapeutic applications for inhibitors and activators NATURE REVIEWS DRUG DISCOVERY Volume: 7 Issue: 2 Pages: 168-181 Published: FEB 2008
    Innocenti, A (Innocenti, Alessio)[ 1 ] ; Vullo, D (Vullo, Daniela)[ 1 ] ; Scozzafava, A (Scozzafava, Andrea)[ 1 ] ; Supuran, CT (Supuran, Claudiu T.)[ 1 ] Carbonic anhydrase inhibitors: Interactions of phenols with the 12 catalytically active mammalian isoforms (CA I-XIV) BIOORGANIC & MEDICINAL CHEMISTRY LETTERS Volume: 18 Issue: 5 Pages: 1583-1587 , 2008
    Innocenti, A (Innocenti, Alessio)[ 1 ] ; Hilvo, M (Hilvo, Mika)[ 2,3 ] ; Scozzafava, A (Scozzafava, Andrea)[ 1 ] ; Lindfors, M (Lindfors, Mikaela)[ 2,3 ] ; Nordlund, HR (Nordlund, Henri R.)[ 2,3 ] ; Kulomaa, MS (Kulomaa, Markku S.)[ 2,3 ] ; Parkkila, S (Parkkila, Seppo)[ 2,3,4 ] ; Supuran, CT Carbonic anhydrase inhibitors: The very weak inhibitors dithiothreitol, beta-mercaptoethanol, tris(carboxyethyl) phosphine and threitol interfere with the binding of sulfonamides to isozymes II and IX IOORGANIC & MEDICINAL CHEMISTRY LETTERS Volume: 18 Issue: 6 Pages: 1898-1903, 2008
    Saczewski, F (Saczewski, Franciszek)[ 1 ] ; Innocenti, A (Innocenti, Alessio)[ 2 ] ; Slawinski, J (Slawinski, Jaroslaw)[ 1 ] ; Kornicka, A (Kornicka, Anita)[ 1 ] ; Brzozowski, Z (Brzozowski, Zdzislaw)[ 1 ] ; Pomarnacka, E (Pomarnacka, Elzbieta)[ 1 ] ; Scozzafava, A (Scozzafava, Andrea)[ 2 ] ; Temperini, C (Temperini, Claudia)[ 2 ] ; Supuran, CT (Supuran, Claudiu T.)[ 2 ] Carbonic anhydrase inhibitors: Inhibition of human cytosolic isozymes I and II and tumor-associated isozymes IX and XII with S-substituted 4-chloro-2-mercapto-5-methyl-benzenesulfonamides IOORGANIC & MEDICINAL CHEMISTRY Volume: 16 Issue: 7 Pages: 3933-3940, 2008
    Guler, O. Ozensoy; Arslan, O.; Kockar, F Differential in vitro inhibitory effects of anticancer drugs on tumor-associated carbonic anhydrase isozymes CA IX and CA XII METHODS AND FINDINGS IN EXPERIMENTAL AND CLINICAL PHARMACOLOGY Volume: 30 Issue: 5 Pages: 335-340 Published: JUN 2008
    Supuran, Claudiu T. evelopment of small molecule carbonic anhydrase IX inhibitors Conference: International Carbonic Anhydrase IX (CAIX) Symposium Location: Brussels, BELGIUM Date: NOV, 2007 BJU INTERNATIONAL Volume: 101 Supplement: 4 Pages: 39-40 Published: JUN 2008
    Thiry, A (Thiry, Anne)[ 1 ] ; Supuran, CT (Supuran, Claudiu T.)[ 2 ] ; Masereel, B (Masereel, Bernard)[ 1 ] ; Dogne, JM (Dogne, Jean-Michel)[ 1 ] Recent developments of carbonic anhydrase inhibitors as potential anticancer drugs OURNAL OF MEDICINAL CHEMISTRY Volume: 51 Issue: 11 Pages: 3051-3056, 2008
    Innocenti, A (Innocenti, Alessio)[ 1 ] ; Maresca, A (Maresca, Alfonso)[ 1 ] ; Scozzafava, A (Scozzafava, Andrea)[ 1 ] ; Supuran, CT (Supuran, Claudiu T.)[ 1 ] Carbonic anhydrase inhibitors: Thioxolone versus sulfonamides for obtaining isozyme-selective inhibitors? BIOORGANIC & MEDICINAL CHEMISTRY LETTERS Volume: 18 Issue: 14 Pages: 3938-3941, 2008
    Said, HM (Said, Harun M.)[ 1 ] ; Polat, B (Polat, Buelent)[ 1 ] ; Staab, A (Staab, Adrian)[ 1 ] ; Hagemann, C (Hagemann, Carsten)[ 2 ] ; Stein, S (Stein, Susanne)[ 3 ] ; Flentje, M (Flentje, Michael)[ 1 ] ; Theobald, M (Theobal Rapid detection of the hypoxia-regulated CA-IX and NDRG1 gene expression in different glioblastoma cells in vitro ONCOLOGY REPORTS Volume: 20 Issue: 2 Pages: 413-419, 2008
    Innocenti, A (Innocenti, Alessio)[ 1 ] ; Vullo, D (Vullo, Daniela)[ 1 ] ; Scozzafava, A (Scozzafava, Andrea)[ 1 ] ; Supuran, CT (Supuran, Claudiu T.)[ 1 ] Carbonic anhydrase inhibitors: Inhibition of mammalian isoforms I-XIV with a series of substituted phenols including paracetamol and salicylic acid BIOORGANIC & MEDICINAL CHEMISTRY Volume: 16 Issue: 15 Pages: 7424-7428, 2008
    Choi, SW (Choi, Sung-Weon)[ 2 ] ; Kim, JY (Kim, Joo-Young)[ 2 ] ; Park, JY (Park, Joo-Yong)[ 2 ] ; Cha, IH (Cha, In-Ho)[ 3 ] ; Kim, J (Kim, Jin)[ 4 ] ; Lee, S (Lee, Sun)[ 1 ] Expression of carbonic anhydrase IX is associated with postoperative recurrence and poor prognosis in surgically treated oral squamous cell carcinomas HUMAN PATHOLOGY olume: 39 Issue: 9 Pages: 1317-1322, 2008
    Guzel, O (Guezel, Oezlen)[ 1,2 ] ; Innocenti, A (Innocenti, Alessio)[ 1 ] ; Scozzafava, A (Scozzafava, Andrea)[ 1 ] ; Salman, A (Salman, Aydin)[ 2 ] ; Parkkila, S (Parkkila, Seppo)[ 3,4,5 ] ; Hilvo, M (Hilvo, Mika)[ 3,4,5 ] ; Supuran, CT (Supuran, Claudiu T.)[ 1 ] Carbonic anhydrase inhibitors: Synthesis and inhibition studies against mammalian isoforms I-XV with a series of 2-(hydrazinocarbonyl)-3-substituted-phenyl-1H-indole-5-sulfonamides IOORGANIC & MEDICINAL CHEMISTRY Volume: 16 Issue: 20 Pages: 9113-9120, 2008
    Guzel, O (Guzel, Ozlen)[ 1,2 ] ; Innocenti, A (Innocenti, Alessio)[ 1 ] ; Hall, RA (Hall, Rebecca A.)[ 3 ] ; Scozzafava, A (Scozzafava, Andrea)[ 1 ] ; Muhlschlegel, FA (Muhlschlegel, Fritz A.)[ 3 ] ; Supuran, CT (Supuran, Claudiu T.)[ 1 ] Carbonic anhydrase inhibitors. The nematode alpha-carbonic anhydrase of Caenorhabditis elegans CAH-4b is highly inhibited by 2-(hydrazinocarbonyl)-3-substituted-phenyl-1H-indole-5-sulfonamides BIOORGANIC & MEDICINAL CHEMISTRY Volume: 17 Issue: 8 Pages: 3212-3215 , 2009
    Supuran, CT (Supuran, Claudiu T.)[ 2 ] ; Di Fiore, A (Di Fiore, Anna)[ 1 ] ; Alterio, V (Alterio, Vincenzo)[ 1 ] ; Monti, SM (Monti, Simona Maria)[ 1 ] ; De Simone, G (De Simone, Giuseppina)[ 1 ] Recent Advances in Structural Studies of the Carbonic Anhydrase Family: The Crystal Structure of Human CA IX and CA XIII CURRENT PHARMACEUTICAL DESIGN Volume: 16 Issue: 29 Pages: 3246-3254, 2010
    De Simone, G (De Simone, Giuseppina)[ 2 ] ; Supuran, CT (Supuran, Claudiu T.)[ 1 ] Carbonic anhydrase IX: Biochemical and crystallographic characterization of a novel antitumor target OCHIMICA ET BIOPHYSICA ACTA-PROTEINS AND PROTEOMICS Volume: 1804 Issue: 2 Pages: 404-409 Special Issue: SI, 2010
    Pacchiano, F (Pacchiano, Fabio)[ 3 ] ; Carta, F (Carta, Fabrizio)[ 3 ] ; McDonald, PC (McDonald, Paul C.)[ 1,2 ] ; Lou, YM (Lou, Yuanmei)[ 1,2 ] ; Vullo, D (Vullo, Daniela)[ 3 ] ; Scozzafava, A (Scozzafava, Andrea)[ 3 ] ; Dedhar, S (Dedhar, Shoukat)[ 1,2,4 ] ; Supuran, CT (Supuran, Claudiu T.)[ 3 ] Ureido-Substituted Benzenesulfonamides Potently Inhibit Carbonic Anhydrase IX and Show Antimetastatic Activity in a Model of Breast Cancer Metastasis JOURNAL OF MEDICINAL CHEMISTRY Volume: 54 Issue: 6 Pages: 1896-1902, 2011
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    Rami, M (Rami, Marouan)[ 1 ] ; Maresca, A (Maresca, Alfonso)[ 2 ] ; Smaine, FZ (Smaine, Fatma-Zhora)[ 1,3 ] ; Montero, JL (Montero, Jean-Louis)[ 1 ] ; Scozzafava, A (Scozzafava, Andrea)[ 2 ] ; Winum, JY (Winum, Jean-Yves)[ 1 ] ; Supuran, CT (Supuran, Claudiu T.)[ 2 ] Sulfonamides incorporating boroxazolidone moieties are potent inhibitors of the transmembrane, tumor-associated carbonic anhydrase isoforms IX and XII BIOORGANIC & MEDICINAL CHEMISTRY LETTERS Volume: 21 Issue: 10 Pages: 2975-2979, 2011
    Carta, F (Carta, Fabrizio)[ 2 ] ; Garaj, V (Garaj, Vladimir)[ 2,3 ] ; Maresca, A (Maresca, Alfonso)[ 2 ] ; Wagner, J (Wagner, Jason)[ 1 ] ; Avvaru, BS (Avvaru, Balendu Sankara)[ 1 ] ; Robbins, AH (Robbins, Arthur H.)[ 1 ] ; Scozzafava, A (Scozzafava, Andrea)[ 2 ] ; McKenna, R (McKenna, Robert)[ 1 ] ; Supuran, CT (Supuran, Claudiu T.)[ 2 ] Sulfonamides incorporating 1,3,5-triazine moieties selectively and potently inhibit carbonic anhydrase transmembrane isoforms IX, XII and XIV over cytosolic isoforms I and II: Solution and X-ray crystallographic studies BIOORGANIC & MEDICINAL CHEMISTRY Volume: 19 Issue: 10 Pages: 3105-3119, 2011
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    Marushima, H (Marushima, Hideki)[ 1,4 ] ; Shibata, SI (Shibata, Shun-Ichi)[ 1 ] ; Asakura, T (Asakura, Tadashi)[ 1 ] ; Matsuura, T (Matsuura, Tomokazu)[ 2 ] ; Maehashi, H (Maehashi, Haruka)[ 2 ] ; Ishii, Y (Ishii, Yuji)[ 4 ] ; Eda, H (Eda, Homare)[ 1 ] ; Aoki, K (Aoki, Katsuhiko)[ 1 ] ; Iida, Y (Iida, Yasushi)[ 3 ] ; Morikawa, T (Morikawa, Toshiaki)[ 4 ] ; Ohkawa, K Three-dimensional culture promotes reconstitution of the tumor-specific hypoxic microenvironment under TGF beta stimulation INTERNATIONAL JOURNAL OF ONCOLOGY Volume: 39 Issue: 5 Pages: 1327-1336, 2011
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    KRYMOV, S.K. - SCHERBAKOV, A.M. - DEZHENKOVA, L.G. - SALNIKOVA, D.I. - SOLOV'EVA, S.E. - SOROKIN, D.V. - VULLO, D. - DE LUCA, V. - CAPASSO, C. - SUPURAN, C.T. - SHCHEKOTIKHIN, A.E. Indoline-5-Sulfonamides: A Role of the Core in Inhibition of Cancer-Related Carbonic Anhydrases, Antiproliferative Activity and Circumventing of Multidrug Resistance. In PHARMACEUTICALS. DEC 2022, vol. 15, no. 12.
    SUPURAN, Claudiu T. Targeting carbonic anhydrases for the management of hypoxic metastatic tumors. In EXPERT OPINION ON THERAPEUTIC PATENTS. ISSN 1354-3776, NOV 2 2023, vol. 33, no. 11, SI, p. 701-720. Dostupné na: https://doi.org/10.1080/13543776.2023.2245971.
    KategóriaABC - Kapitoly vo vedeckých monografiách vydané v zahraničných vydavateľstvách
    Kategória (od 2022)V2 - Vedecký výstup publikačnej činnosti ako časť editovanej knihy alebo zborníka
    Typ výstupukapitola
    Rok vykazovania2004
    Registrované vCCC
    článok

    článok

    rokCCIFIF Q (best)JCR Av Jour IF PercSJRSJR Q (best)CiteScore
    A
    rok vydaniarok metrikyIFIF Q (best)SJRSJR Q (best)
    2004
Počet záznamov: 1  

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