Počet záznamov: 1  

Structure-activity relations on [1-(3,5-difluoro-4-hydroxyphenyl)-1H-pyrrol-3-yl]phenylmethanone. The effect of methoxy substitution on aldose reductase inhibitory activity and selectivity

  1. NázovStructure-activity relations on [1-(3,5-difluoro-4-hydroxyphenyl)-1H-pyrrol-3-yl]phenylmethanone. The effect of methoxy substitution on aldose reductase inhibitory activity and selectivity
    Autor Chatzopoulou Maria
    Spoluautori Mamadou Eduard

    Jusková Mária 1983- SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV    SCOPUS    SCOPUS

    Koukoulitsa Cathrine

    Nicolaou Ioannis

    Štefek Milan 1950-2023 SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV    SCOPUS    ORCID

    Demopoulos Vassilis J.

    Zdroj.dok. Bioorganic & Medicinal Chemistry. Vol. 19, no. 4 (2011), p. 1426-1433
    Jazyk dok.eng - angličtina
    KrajinaGB - Veľká Británia
    Druh dok.rozpis článkov z periodík (rbx)
    OhlasyZANATTA, N. - AQUINO, E.D. - DA SILVA, F.M. - BONACORSO, H.G. - MARTINS, M.A.P. Improved One-Pot Synthesis of 1-Aryl-3-trifluoroacetyl-1H-pyrroles under Swern Oxidation. In SYNTHESIS-STUTTGART. ISSN 0039-7881, 2012, vol. 44, no. 22, p. 3477-3482.
    ALI, S. - SAEED, A. - ABBAS, N. - SHAHID, M. - BOLTE, M. - IQBAL, J. Design, synthesis and molecular modelling of novel methyl[4-oxo-2-(aroylimino)-3-(substituted phenyl)thiazolidin-5-ylidene]acetates as potent and selective aldose reductase inhibitors. In MEDCHEMCOMM. ISSN 2040-2503, 2012, vol. 3, no. 11, p. 1428-1434.
    IQBAL, Z. - ALI, S. - IQBAL, J. - ABBAS, Q. - QURESHI, I.Z. - HAMEED, S. Dual action spirobicycloimidazolidine-2,4-diones: Antidiabetic agents and inhibitors of aldose reductase-an enzyme involved in diabetic complications. In BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. ISSN 0960-894X, 2013, vol. 23, no. 2, p. 488-491.
    POSTIKOVA, S. - SABBAH, M. - WIGHTMAN, D. - NGUYEN, I.T. - SANSELME, M. - BESSON, T. - BRIERE, J.F. - OUDEYER, S. - LEVACHER, V. Developments in Meyers' Lactamization Methodology: En Route to Bi(hetero)aryl Structures with Defined Axial Chirality. In JOURNAL OF ORGANIC CHEMISTRY. ISSN 0022-3263, 2013, vol. 78, no. 16, p. 8191-8197.
    REDDY, T. N. - RAVINDER, M. - BAGUL, P. - RAVIKANTI, K. - BAGUL, Ch. - NANUBOLU, J. B. - SRINIVAS, K. - BANERJEE, S. K. - RAO, V. J. Synthesis and biological evaluation of new epalrestat analogues as aldose reductase inhibitors (ARIs). In EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. ISSN 0223-5234; 1768-3254, 2014, vol. 71, p. 53-66.
    OVAIS, S. - PUSHPALATHA, H. - REDDY, G. B. - RATHORE, P. - BASHIR, R. - YASEEN, S. - DHEYAA, A. - YASEEN, R. - TANWAR, O. - AKTHAR, M. - SAMIM, M. - JAVED, K. Synthesis and biological evaluation of some new pyrazoline substituted benzenesulfonylurea/thiourea derivatives as anti-hyperglycaemic agents and aldose reductase inhibitors. In EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. ISSN 0223-5234; 1768-3254, 2014, vol. 80, p. 209-217.
    MACCARI, R. - OTTANA, R. Targeting aldose reductase for the treatment of diabetes complications and inflammatory diseases: New insights and future directions. In JOURNAL OF MEDICINAL CHEMISTRY. ISSN 0022-2623, 2015, vol. 58, no. 5, p. 2047-2067.
    ZOU, Y. - QIN, X.Y. - HAO, X. - ZHANG, W. - YANG, S.Q. - YANG, Y.C. - HAN, Z.F. - MA, B. - ZHU, C.J. Phenolic 4-hydroxy and 3,5-dihydroxy derivatives of 3-phenoxyquinoxalin-2(1H)-one as potent aldose reductase inhibitors with antioxidant activity. In BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS. ISSN 0960-894X, 2015, vol. 25, no. 18, p. 3924-3927.
    PLIOUKAS, M. - GABRIELI, C. - LAZARI, D. - KOKKALOU, E. Phytochemical analysis with the antioxidant and aldose reductase inhibitory capacities of Tephrosia humilis aerial parts' extracts. In NATURAL PRODUCT RESEARCH. ISSN 1478-6419, 2016, vol. 30, no. 12, p. 1366-1372.
    SUNKE, R. - NALLAPATI, S.B. - KUMAR, J.S. - KUMAR, K.S. - PAL, M. Use of AlCl3 in Friedel Crafts arylation type reactions and beyond: an overview on the development of unique methodologies leading to N-heteroarenes. In ORGANIC & BIOMOLECULAR CHEMISTRY. ISSN 1477-0520, 2017, vol. 15, no. 19, p. 4042-4057.
    ZHAN, J.-Y. - MA, K. - ZHENG, Q.-C. - YANG, G.-H. - ZHANG, H.-X. Exploring the interactional details between aldose reductase (AKR1B1) and 3-Mercapto-5H-1,2,4-triazino[5,6-b]indole-5-acetic acid through molecular dynamics simulations. In JOURNAL OF BIOMOLECULAR STRUCTURE & DYNAMICS. ISSN 0739-1102, 2019, vol. 37, no. 7, p. 1724-1735.
    HAO, Xin - QI, Gang - MA, Hongxing - ZHU, Changjin - HAN, Zhongfei. Novel 2-phenoxypyrido[3,2-b]pyrazin-3(4H)-one derivatives as potent and selective aldose reductase inhibitors with antioxidant activity. In JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY. ISSN 1475-6366, 2019, vol. 34, no. 1, pp. 1368-1372.
    HAO, X. - QIN, X.Y. - ZHANG, X. - MA, B. - QI, G. - YU, T.M. - HAN, Z.F. - ZHU, C.J. Identification of quinoxalin-2(1H)-one derivatives as a novel class of multifunctional aldose reductase inhibitors. In FUTURE MEDICINAL CHEMISTRY. ISSN 1756-8919, DEC 2019, vol. 11, no. 23, p. 2989-3004.
    MOUSSOUNI, S. - KARAKOUSI, C.V. - TSATALAS, P. - LAZARI, D. - KOKKALOU, E. Biological Studies with Phytochemical Analysis Of Cornus mas Unripe Fruits. In CHEMISTRY OF NATURAL COMPOUNDS. ISSN 0009-3130, 2020, vol. 56, no. 1.
    KUMAR, M. - CHOUDHARY, S. - SINGH, P.K. - SILAKARI, O. Addressing selectivity issues of aldose reductase 2 inhibitors for the management of diabetic complications. In FUTURE MEDICINAL CHEMISTRY. ISSN 1756-8919, 2020, vol. 12, no. 14, p. 1327-1358.
    KategóriaADCA - Vedecké práce v zahraničných karentovaných časopisoch impaktovaných
    Kategória (od 2022)V3 - Vedecký výstup publikačnej činnosti z časopisu
    Typ výstupučlánok
    Rok vykazovania2011
    Registrované vWOS
    Registrované vSCOPUS
    Registrované vCCC
    DOI 10.1016/j.bmc.2011.01.009
    článok

    článok

    rokCCIFIF Q (best)JCR Av Jour IF PercSJRSJR Q (best)CiteScore
    A
    rok vydaniarok metrikyIFIF Q (best)SJRSJR Q (best)
    201120102.978Q21.083Q1
Počet záznamov: 1  

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