Počet záznamov: 1  

Decreasing acidity in a series of aldose reductase inhibitors: 2-Fluoro-4-(1H-pyrrol-1-yl)phenol as a scaffold for improved membrane permeation

  1. NázovDecreasing acidity in a series of aldose reductase inhibitors: 2-Fluoro-4-(1H-pyrrol-1-yl)phenol as a scaffold for improved membrane permeation
    Autor Chatzopoulou Maria
    Spoluautori Patsilinakos Alexandros

    Vallianatou Theodosia

    Šoltésová Prnová Marta 1986- SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV    SCOPUS    ORCID

    Žakelj Simon

    Ragno Rino

    Štefek Milan 1950-2023 SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV    SCOPUS    ORCID

    Kristl Albin

    Tsantili-Kakoulidou Anna

    Demopoulos Vassilis J.

    Zdroj.dok. Bioorganic & Medicinal Chemistry. Vol. 22 (2014), p. 2194-2207
    Jazyk dok.eng - angličtina
    KrajinaGB - Veľká Británia
    Druh dok.rozpis článkov z periodík (rbx)
    OhlasyPEREZ, W.I. - SOTO, Y. - ORTIZ, C. - MATTA, J. - MELENDEZ, E. Ferrocenes as potential chemotherapeutic drugs: Synthesis, cytotoxic activity, reactive oxygen species production and micronucleus assay. In BIOORGANIC & MEDICINAL CHEMISTRY. ISSN 0968-0896, 2015, vol. 23, no. 3, p. 471-479.
    MACCARI, R. - OTTANA, R. Targeting aldose reductase for the treatment of diabetes complications and inflammatory diseases: New insights and future directions. In JOURNAL OF MEDICINAL CHEMISTRY. ISSN 0022-2623, 2015, vol. 58, no. 5, p. 2047-2067.
    PEREZ W.I. - RHEINGOLD A.L. - MELENDEZ E. Crystal structure of bis[4-(1H-pyrrol-1-yl) phenyl]ferrocene-1,1´-dicarboxylate: a potential chemotherapeutic drug. In ACTA CRYSTALLOGRAPHICA, SECTION E. ISSN 2056-9890, 2015, vol. 71, part 5, p. 536-539.
    GREWAL, A.S. - BHARDWAJ, S. - PANDITA, D. - LATHER, V. - SEKHON, B.S. Updates on Aldose Reductase Inhibitors for Management of Diabetic Complications and Non-diabetic Diseases. In MINI-REVIEWS IN MEDICINAL CHEMISTRY. ISSN 1389-5575, 2016, vol. 16, no. 2, p. 120-162.
    GHOLAP, S.S. Pyrrole: An emerging scaffold for construction of valuable therapeutic agents. In EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. ISSN 0223-5234, 2016, vol. 110, p. 13-31.
    MAGALHAES, F.E.A. - BATISTA, F.L.A. - SERPA, O.F. - MOURA, L.F.W.G. - LIMA, M.D.L. - DA SILVA, A.R.A. - GUEDES, M.I.F. - SANTOS, S.A.A.R. - DE OLIVEIRA, B.A. - NOGUEIRA, A.B. - BARBOSA, T.M. - HOLANDA, D.K.R. - DAMASCENO, M.B.M.V. - DE MELO, J.D.A. - BARROSO, L.K.V. - CAMPOS, A.R. Orofacial antinociceptive effect of Mimosa tenuiflora (Willd.) Poiret. In BIOMEDICINE & PHARMACOTHERAPY. ISSN 0753-3322, 2018, vol. 97, p. 1575-1585.
    KERRU, N. - SINGH-PILLAY, A. - AWOLADE, P. - SINGH, P. Current anti-diabetic agents and their molecular targets: A review. In EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. ISSN 0223-5234, 2018, vol. 152, p. 436-488.
    ALFORD, M.A. - TIAN, Z. - MENARD, F. - KLEGERIS, A. Characterization of novel kainic acid analogs as inhibitors of select microglial functions. In EUROPEAN JOURNAL OF PHARMACOLOGY. ISSN 0014-2999, 2019, vol. 851, p. 25-35.
    DOWARAH, J. - SINGH, V.P. Anti-diabetic drugs recent approaches and advancements. In BIOORGANIC & MEDICINAL CHEMISTRY. ISSN 0968-0896, 2020, vol. 28, no. 5.
    HAN, Z.F. - ZHU, J.K. - ZHANG, Y.N. - ZHANG, Y. - ZHANG, H.Y. - QI, G. - ZHU, C.J. - HAO, X. Novel quinolin-4(1H)-one derivatives as multi-effective aldose reductase inhibitors for treatment of diabetic complications: Synthesis, biological evaluation, and molecular modeling studies. In BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. ISSN 0960-894X, 2020, vol. 30, no. 9, art. no. 127101.
    KOUSAXIDIS, A. - PETROU, A. - LAVRENTAKI, V. - FESATIDOU, M. - NICOLAOU, I. - GERONIKAKI, A. Aldose reductase and protein tyrosine phosphatase 1B inhibitors as a promising therapeutic approach for diabetes mellitus. In EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. ISSN 0223-5234, DEC 1 2020, vol. 207.
    RUIZ, Francesc Xavier - PARES, Xavier - FARRES, Jaume. Perspective on the Structural Basis for Human Aldo-Keto Reductase 1B10 Inhibition. In METABOLITES, 2021, vol. 11, no. 12, pp. Dostupné na: https://doi.org/10.3390/metabo11120865.
    HAJLAOUI, A. - ASSEL, A. - LAZRAG, H. - BOUAJILA, J. - HARRATH, A.H. - MANSOUR, L. - JANNET, H.B. - ROMDHANE, A. Design, Synthesis and biological evaluation of novel benzopyran derivatives as potential alpha-amylase inhibitors: An Investigation by Experimental and Computational Studies. In JOURNAL OF MOLECULAR STRUCTURE. ISSN 0022-2860, FEB 5 2023, vol. 1273. Dostupné na: https://doi.org/10.1016/j.molstruc.2022.134227.
    GANESH, B.H. - RAJ, A.G. - ARUCHAMY, B. - NANJAN, P. - DRAGO, C. - RAMANI, P. Pyrrole: A Decisive Scaffold for the Development of Therapeutic Agents and Structure-Activity Relationship. In CHEMMEDCHEM. ISSN 1860-7179, JAN 2 2024, vol. 19, no. 1. Dostupné na: https://doi.org/10.1002/cmdc.202300447.
    KategóriaADCA - Vedecké práce v zahraničných karentovaných časopisoch impaktovaných
    Kategória (od 2022)V3 - Vedecký výstup publikačnej činnosti z časopisu
    Typ výstupučlánok
    Rok vykazovania2014
    Registrované vWOS
    Registrované vSCOPUS
    Registrované vCCC
    DOI 10.1016/j.bmc.2014.02.016
    článok

    článok

    Názov súboruPrístupVeľkosťStiahnutéTypLicence
    Decreasing acidity in a series of aldose reductase inhibitors....pdfNeprístupný/archív2.1 MB1Vydavateľská verzia
    rokCCIFIF Q (best)JCR Av Jour IF PercSJRSJR Q (best)CiteScore
    A
    rok vydaniarok metrikyIFIF Q (best)SJRSJR Q (best)
    201420132.951Q21.063Q1
Počet záznamov: 1  

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