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Identification of novel aldose reductase inhibitors based on carboxymethylated mercaptotriazinoindole scaffold
Názov Identification of novel aldose reductase inhibitors based on carboxymethylated mercaptotriazinoindole scaffold Autor Štefek Milan 1950-2023 SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV SCOPUS ORCID Spoluautori Šoltésová Prnová Marta 1986- SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV SCOPUS ORCID Májeková Magdaléna 1958- SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV SCOPUS RID ORCID Rechlin Chris Heine Andreas Klebe Gerhard Zdroj.dok. Journal of Medicinal Chemistry. Vol. 58, no. 6 (2015), p. 2649-2657 Jazyk dok. eng - angličtina Krajina US - Spojené štáty Druh dok. rozpis článkov z periodík (rbx) Ohlasy ANTONY P. - VIJAYAN R. Identification of Novel Aldose Reductase Inhibitors from Spices: A Molecular Docking and Simulation Study. IN PLOS ONE. ISSN 1932-6203 (Electronic), 2015, vol. 10, no. 9, art. no. e0138186. 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ISSN 2046-2069, 2017, vol. 7, no. 15, p. 9264-9271. EL-SAYED, S. - METWALLY, K. - EL-SHANAWANI, A.A. - ABDEL-AZIZ, L.M. - EL-RASHEDY, A.A. - SOLIMAN, M.E.S. - QUATTRINI, L. - COVIELLO, V. - LA MOTTA, C. Quinazolinone-based rhodanine-3-acetic acids as potent aldose reductase inhibitors: Synthesis, functional evaluation and molecular modeling study. In BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS. ISSN 0960-894X, 2017, vol. 27, no. 20, p. 4760-4764. METWALLY, K. - PRATSINIS, H. - KLETSAS, D. - QUATTRINI, L. - COVIELLO, V. - LA MOTTA, C. - EL-RASHEDY, A.A. - SOLIMAN, M.E.S. Novel quinazolinone-based 2,4-thiazolidinedione-3-acetic acid derivatives as potent aldose reductase inhibitors. In FUTURE MEDICINAL CHEMISTRY. ISSN 1756-8919, 2017, vol. 9, no. 18, p. 2147-2166. SOBEH, M. - MAHMOUD, M.F. - ABDELFATTAH, M.A.O. - EL-BESHBISHY, H.A. - EL-SHAZLY, A.M. - WINK, M. Albizia harveyi: phytochemical profiling, antioxidant, antidiabetic and hepatoprotective activities of the bark extract. 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ISSN 0960-894X, 2020, vol. 30, no. 9, art. no. 127101. KOUSAXIDIS, A. - PETROU, A. - LAVRENTAKI, V. - FESATIDOU, M. - NICOLAOU, I. - GERONIKAKI, A. Aldose reductase and protein tyrosine phosphatase 1B inhibitors as a promising therapeutic approach for diabetes mellitus. In EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. ISSN 0223-5234, DEC 1 2020, vol. 207, art. no. 112742. KUMAR, M. - CHOUDHARY, S. - SINGH, P.K. - SILAKARI, O. Addressing selectivity issues of aldose reductase 2 inhibitors for the management of diabetic complications. In FUTURE MEDICINAL CHEMISTRY. ISSN 1756-8919, 2020, vol. 12, no. 14, p. 1327-1358. SONOWAL, H. - RAMANA, K.V. Development of Aldose Reductase Inhibitors for the Treatment of Inflammatory Disorders and Cancer: Current Drug Design Strategies and Future Directions. In CURRENT MEDICINAL CHEMISTRY. ISSN 0929-8673, 2021, vol. 28, no. 19, p. 3683-3712. ZHU, Junkai - QI, Gang - KUANG, Yan - ZHAO, Yating - SUN, Xinjie - ZHU, Changjin - HAO, Xin - HAN, Zhongfei. Identification of 9H-purin-6-amine derivatives as novel aldose reductase inhibitors for the treatment of diabetic complications. In ARCHIV DER PHARMAZIE, 2022, vol. 355, no. 8, pp. ISSN 0365-6233. Dostupné na: https://doi.org/10.1002/ardp.202200043. YAHYA, S. - HAIDER, K. - PATHAK, A. - CHOUDHARY, A. - HOODA, P. - SHAFEEQ, M. - YAR, M.S. Strategies in synthetic design and structure-activity relationship studies of novel heterocyclic scaffolds as aldose reductase-2 inhibitors. In ARCHIV DER PHARMAZIE. ISSN 0365-6233, DEC 2022, vol. 355, no. 12. Dostupné na: https://doi.org/10.1002/ardp.202200167. TASSOPOULOU, V.P. - TZARA, A. - KOUROUNAKIS, A.P. Design of Improved Antidiabetic Drugs: A Journey from Single to Multitarget Agents. In CHEMMEDCHEM. ISSN 1860-7179, DEC 5 2022, vol. 17, no. 23. Dostupné na: https://doi.org/10.1002/cmdc.202200320. PANAGIOTIS, Theodosis Nobelos - STAVROS, Kokkinos - CHARALAMPOS, Triantis. Diabetes in Alzheimer disease Interaction at mechanistic and therapeutic level. In Pharmakeftiki, 2022-01-01, 34, 3, pp. 103-117. ISSN 11054999. HAN, Zhongfei - LI, Jiahui - XU, Zilu - SU, Yu - WANG, Yihan - ZHUO, Lili - DU, Jiaming - ZHU, Changjin - HAO, Xin. Design and synthesis of novel quinazolin-4(1H)-one derivatives as potent and selective inhibitors targeting AKR1B1. In ARCHIV DER PHARMAZIE, 2023, vol. 356, no. 4, pp. ISSN 0365-6233. Dostupné na: https://doi.org/10.1002/ardp.202200577. PATNAM, N. - CHEVULA, K. - CHENNAMSETTI, P. - KRAMADHATI, S. - ALAPARTHI, M.D. - MANGA, V. Novel thiazolidinedione (TZD) scaffolds as aldose reductase inhibitors, synthesis and molecular docking studies. In CHEMICAL DATA COLLECTIONS. AUG 2023, vol. 46. Dostupné na: https://doi.org/10.1016/j.cdc.2023.101045. ALSHAGHDALI, K. - ALHARAZI, T. - REZGUI, R. - ACAR, T. - ALJERWAN, R.F. - ALTAYYAR, A. - TASLEEM, M. - SAEED, M. - YADAV, D.K. - SAEED, A. Identification and evaluation of putative type 2 diabetes mellitus inhibitors derived from Cichorium intybus. In JOURNAL OF MOLECULAR STRUCTURE. ISSN 0022-2860, JUN 15 2024, vol. 1306. Dostupné na: https://doi.org/10.1016/j.molstruc.2024.137629. KUMARI, P. - KOHAL, R. - BHAVANA - GUPTA, G.D. - VERMA, S.K. Selectivity challenges for aldose reductase inhibitors: A review on comparative SAR and interaction studies. In JOURNAL OF MOLECULAR STRUCTURE. ISSN 0022-2860, DEC 15 2024, vol. 1318, 1. Dostupné na: https://doi.org/10.1016/j.molstruc.2024.139207. PATNAM, N. - CHEVULA, K. - CHENNAMSETTI, P. - ALETI, B. - KOTHA, A.K. - MANGA, V. Synthesis, antidiabetic activity and molecular docking studies of novel aryl benzylidenethiazolidine-2,4-dione based 1,2,3-triazoles. In MOLECULAR DIVERSITY. ISSN 1381-1991, JUN 2024, vol. 28, no. 3, p. 1551-1563. Dostupné na: https://doi.org/10.1007/s11030-023-10674-y. Kategória ADCA - Vedecké práce v zahraničných karentovaných časopisoch impaktovaných Kategória (od 2022) V3 - Vedecký výstup publikačnej činnosti z časopisu Typ výstupu článok Rok vykazovania 2015 Registrované v WOS Registrované v SCOPUS Registrované v CCC DOI 10.1021/jm5015814 
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Názov súboru Prístup Veľkosť Stiahnuté Typ Licence Identification of novel aldose reductase inhibitors based on carboxymethylated....pdf Neprístupný/archív 2.2 MB 1 Vydavateľská verzia rok CC IF IF Q (best) JCR Av Jour IF Perc SJR SJR Q (best) CiteScore A rok vydania rok metriky IF IF Q (best) SJR SJR Q (best) 2015 2014 5.447 Q1 2.240 Q1
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