Počet záznamov: 1  

Identification of novel aldose reductase inhibitors based on carboxymethylated mercaptotriazinoindole scaffold

  1. NázovIdentification of novel aldose reductase inhibitors based on carboxymethylated mercaptotriazinoindole scaffold
    Autor Štefek Milan 1950-2023 SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV    SCOPUS    ORCID
    Spoluautori Šoltésová Prnová Marta 1986- SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV    SCOPUS    ORCID

    Májeková Magdaléna 1958- SAVEXFATO - Ústav experimentálnej farmakológie a toxikológie SAV    SCOPUS    RID    ORCID

    Rechlin Chris

    Heine Andreas

    Klebe Gerhard

    Zdroj.dok. Journal of Medicinal Chemistry. Vol. 58, no. 6 (2015), p. 2649-2657
    Jazyk dok.eng - angličtina
    KrajinaUS - Spojené štáty
    Druh dok.rozpis článkov z periodík (rbx)
    OhlasyANTONY P. - VIJAYAN R. Identification of Novel Aldose Reductase Inhibitors from Spices: A Molecular Docking and Simulation Study. IN PLOS ONE. ISSN 1932-6203 (Electronic), 2015, vol. 10, no. 9, art. no. e0138186.
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    GOPINATH, G. - SANKESHI, V. - PERUGU, S. - ALAPARTHI, M.D. - BANDARU, S. - PASALA, V.K. - CHITTINENI, P.R. - KRUPADANAM, G.L.D. - SAGURTHI, S.R. Design and synthesis of chiral 2H-chromene-N-imidazolo-amino acid conjugates as aldose reductase inhibitors. In EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. ISSN 0223-5234, 2016, vol. 124, p. 750-762.
    ZHAO, H.W. - PANG, H.L. - ZHAO, Y.D. - LIU, Y.Y. - ZHAO, L.J. - CHEN, X.Q. - SONG, X.Q. - FENG, N.N. - DU, J. Construction of 2,3,4,5-tetrahydro-1,2,4-triazines via [4 + 2] cycloaddition of α-halogeno hydrazones to imines. In RSC ADVANCES. ISSN 2046-2069, 2017, vol. 7, no. 15, p. 9264-9271.
    EL-SAYED, S. - METWALLY, K. - EL-SHANAWANI, A.A. - ABDEL-AZIZ, L.M. - EL-RASHEDY, A.A. - SOLIMAN, M.E.S. - QUATTRINI, L. - COVIELLO, V. - LA MOTTA, C. Quinazolinone-based rhodanine-3-acetic acids as potent aldose reductase inhibitors: Synthesis, functional evaluation and molecular modeling study. In BIOORGANIC AND MEDICINAL CHEMISTRY LETTERS. ISSN 0960-894X, 2017, vol. 27, no. 20, p. 4760-4764.
    METWALLY, K. - PRATSINIS, H. - KLETSAS, D. - QUATTRINI, L. - COVIELLO, V. - LA MOTTA, C. - EL-RASHEDY, A.A. - SOLIMAN, M.E.S. Novel quinazolinone-based 2,4-thiazolidinedione-3-acetic acid derivatives as potent aldose reductase inhibitors. In FUTURE MEDICINAL CHEMISTRY. ISSN 1756-8919, 2017, vol. 9, no. 18, p. 2147-2166.
    SOBEH, M. - MAHMOUD, M.F. - ABDELFATTAH, M.A.O. - EL-BESHBISHY, H.A. - EL-SHAZLY, A.M. - WINK, M. Albizia harveyi: phytochemical profiling, antioxidant, antidiabetic and hepatoprotective activities of the bark extract. In MEDICINAL CHEMISTRY RESEARCH. ISSN 1054-2523, 2017, vol. 26, no. 12, p. 3091-3105.
    YU, J. - CAI, C. Photocatalytic oxidative cyclization of Α-halo hydrazones with tetrahydroisoquinoline for construction of isoquino[3,4-a][1,2,4]-triazines. In CATALYSIS COMMUNICATIONS. ISSN 1566-7367, 2018, vol. 109, p. 60-64.
    ZHANG, C.L. - LI, Y.Z. - LI, J.Y. - LI, Y.L. - GONG, R.Q. - WANG, H.Y. Synthesis and Bioactivities of Novel 1,2,4-Triazine Scheleton Phenanthroline Derivatives and the Fluorescent Recognition on DNA Using Three Novel Co(III) Complexes. In CHINESE JOURNAL OF ORGANIC CHEMISTRY. ISSN 0253-2786, 2018, vol. 38, no. 10, p. 2720-2730.
    ZHAN, J.Y. - MA, K. - ZHENG, Q.C. - YANG, G.H. - ZHANG, H.X. Exploring the interactional details between aldose reductase (AKR1B1) and 3-Mercapto-5H-1,2,4-triazino[5,6-b]indole-5-acetic acid through molecular dynamics simulations. In JOURNAL OF BIOMOLECULAR STRUCTURE & DYNAMICS. ISSN 0739-1102, 2019, vol. 37, no. 7, p. 1724-1735.
    SOBEH, M. - EL-RAEY, M. - REZQ, S. - ABDELFATTAH, M.A.O. - PETRUK, G. - OSMAN, S. - EL-SHAZLY, A.M. - EL-BESHBISHY, H.A. - MAHMOUD, M.F. - WINK, M. Chemical profiling of secondary metabolites of Eugenia uniflora and their antioxidant, anti-inflammatory, pain killing and anti-diabetic activities: A comprehensive approach. In JOURNAL OF ETHNOPHARMACOLOGY. ISSN 0378-8741, 2019, vol. 240, art. no. 111939.
    YANG, Y. - YANG, Q.H. - YU, J. - WAN, W.C. - WEI, X.Y. Characterization of structural requirement for binding of gigantol and aldose reductase. In FRONTIERS IN BIOSCIENCE-LANDMARK. ISSN 1093-9946, 2019, vol. 24, p. 1024-1036.
    HAN, Z.F. - ZHU, J.K. - ZHANG, Y.N. - ZHANG, Y. - ZHANG, H.Y. - QI, G. - ZHU, C.J. - HAO, X. Novel quinolin-4(1H)-one derivatives as multi-effective aldose reductase inhibitors for treatment of diabetic complications: Synthesis, biological evaluation, and molecular modeling studies. In BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. ISSN 0960-894X, 2020, vol. 30, no. 9, art. no. 127101.
    KOUSAXIDIS, A. - PETROU, A. - LAVRENTAKI, V. - FESATIDOU, M. - NICOLAOU, I. - GERONIKAKI, A. Aldose reductase and protein tyrosine phosphatase 1B inhibitors as a promising therapeutic approach for diabetes mellitus. In EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. ISSN 0223-5234, DEC 1 2020, vol. 207, art. no. 112742.
    KUMAR, M. - CHOUDHARY, S. - SINGH, P.K. - SILAKARI, O. Addressing selectivity issues of aldose reductase 2 inhibitors for the management of diabetic complications. In FUTURE MEDICINAL CHEMISTRY. ISSN 1756-8919, 2020, vol. 12, no. 14, p. 1327-1358.
    SONOWAL, H. - RAMANA, K.V. Development of Aldose Reductase Inhibitors for the Treatment of Inflammatory Disorders and Cancer: Current Drug Design Strategies and Future Directions. In CURRENT MEDICINAL CHEMISTRY. ISSN 0929-8673, 2021, vol. 28, no. 19, p. 3683-3712.
    ZHU, Junkai - QI, Gang - KUANG, Yan - ZHAO, Yating - SUN, Xinjie - ZHU, Changjin - HAO, Xin - HAN, Zhongfei. Identification of 9H-purin-6-amine derivatives as novel aldose reductase inhibitors for the treatment of diabetic complications. In ARCHIV DER PHARMAZIE, 2022, vol. 355, no. 8, pp. ISSN 0365-6233. Dostupné na: https://doi.org/10.1002/ardp.202200043.
    YAHYA, S. - HAIDER, K. - PATHAK, A. - CHOUDHARY, A. - HOODA, P. - SHAFEEQ, M. - YAR, M.S. Strategies in synthetic design and structure-activity relationship studies of novel heterocyclic scaffolds as aldose reductase-2 inhibitors. In ARCHIV DER PHARMAZIE. ISSN 0365-6233, DEC 2022, vol. 355, no. 12. Dostupné na: https://doi.org/10.1002/ardp.202200167.
    TASSOPOULOU, V.P. - TZARA, A. - KOUROUNAKIS, A.P. Design of Improved Antidiabetic Drugs: A Journey from Single to Multitarget Agents. In CHEMMEDCHEM. ISSN 1860-7179, DEC 5 2022, vol. 17, no. 23. Dostupné na: https://doi.org/10.1002/cmdc.202200320.
    PANAGIOTIS, Theodosis Nobelos - STAVROS, Kokkinos - CHARALAMPOS, Triantis. Diabetes in Alzheimer disease Interaction at mechanistic and therapeutic level. In Pharmakeftiki, 2022-01-01, 34, 3, pp. 103-117. ISSN 11054999.
    HAN, Zhongfei - LI, Jiahui - XU, Zilu - SU, Yu - WANG, Yihan - ZHUO, Lili - DU, Jiaming - ZHU, Changjin - HAO, Xin. Design and synthesis of novel quinazolin-4(1H)-one derivatives as potent and selective inhibitors targeting AKR1B1. In ARCHIV DER PHARMAZIE, 2023, vol. 356, no. 4, pp. ISSN 0365-6233. Dostupné na: https://doi.org/10.1002/ardp.202200577.
    PATNAM, N. - CHEVULA, K. - CHENNAMSETTI, P. - KRAMADHATI, S. - ALAPARTHI, M.D. - MANGA, V. Novel thiazolidinedione (TZD) scaffolds as aldose reductase inhibitors, synthesis and molecular docking studies. In CHEMICAL DATA COLLECTIONS. AUG 2023, vol. 46. Dostupné na: https://doi.org/10.1016/j.cdc.2023.101045.
    KategóriaADCA - Vedecké práce v zahraničných karentovaných časopisoch impaktovaných
    Kategória (od 2022)V3 - Vedecký výstup publikačnej činnosti z časopisu
    Typ výstupučlánok
    Rok vykazovania2015
    Registrované vWOS
    Registrované vSCOPUS
    Registrované vCCC
    DOI 10.1021/jm5015814
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    Názov súboruPrístupVeľkosťStiahnutéTypLicence
    Identification of novel aldose reductase inhibitors based on carboxymethylated....pdfNeprístupný/archív2.2 MB1Vydavateľská verzia
    rokCCIFIF Q (best)JCR Av Jour IF PercSJRSJR Q (best)CiteScore
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    201520145.447Q12.240Q1
Počet záznamov: 1  

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