Počet záznamov: 1
Carbonic anhydrase inhibitors: The first selective, membrane-impermeant inhibitors targeting the tumor-associated isozyme IX
Názov Carbonic anhydrase inhibitors: The first selective, membrane-impermeant inhibitors targeting the tumor-associated isozyme IX Autor Pastoreková Silvia 1961 SAVVIR - Virologický ústav SAV ORCID Spoluautori Casini A. Scozzafava A. Vullo D. Pastorek Jaromír 1957- SAVVIR - Virologický ústav SAV Supuran C.T. Zdroj.dok. Bioorganic & Medicinal Chemistry Letters. Vol. 14, no. 4 (2004), p. 869 - 873 Jazyk dok. eng - angličtina Krajina SK - Slovenská republika Druh dok. rozpis článkov z periodík (rbx) Ohlasy Bouchez LC, Dubbaka SR, Turks M, Vogel P JOURNAL OF ORGANIC CHEMISTRY 69 (19): 6413-6418 SEP 17 2004 Poulsen SA, Bornaghi LF, Healy PC Synthesis and structure-activity relationships of novel benzene sulfonamides with potent binding affinity for bovine carbonic anhydrase II BIOORGANIC & MEDICINAL CHEMISTRY LETTERS 15 (24): 5429-5433 DEC 15 2005 Bouchez LC, Turks M, Dubbaka SR, Fonquerne F, Craita C, Laclef S, Vogel P Sulfur dioxide mediated one-pot, four-component synthesis of polyfunctional sulfones and sulfonamides, including medium-ring cyclic derivatives TETRAHEDRON 61 (48): 11473-11487 NOV 28 2005 [Anon] Carbonic anhydrase inhibitors: CA IX selective inhibitors incorporating aromatic or heterocyclic sulfonamide EXPERT OPINION ON THERAPEUTIC PATENTS Volume: 15 Issue: 2 Pages: 233-236 Published: FEB 2005 Mizumori M (Mizumori, Misa), Meyerowitz J (Meyerowitz, Justin), Takeuchi T (Takeuchi, Tetsu), Lim S (Lim, Shu), Lee P (Lee, Paul), Supuran CT (Supuran, Claudiu T.), Guth PH (Guth, Paul H.), Engel E (Engel, Eli), Kaunitz JD (Kaunitz, Jonathan D.), Akiba Y (Akiba, Yasutada) Epithelial carbonic anhydrases facilitate P-CO2 and pH regulation in rat duodenal mucosa JOURNAL OF PHYSIOLOGY-LONDON 573 (3): 827-842 JUN 15 2006 Poulsen SA Direct screening of a dynamic combinatorial library using mass spectrometry JOURNAL OF THE AMERICAN SOCIETY FOR MASS SPECTROMETRY 17 (8): 1074-1080 AUG 2006 Akiba Y (Akiba, Yasutada), Ghayouri S (Ghayouri, Sara), Takeuchi T (Takeuchi, Tetsu), Mizumori M (Mizumori, Misa), Guth PH (Guth, Paul H.), Engel E (Engel, Eli), Swenson ER (Swenson, Erik R.), Kaunitz JD (Kaunitz, Jonathan D.) Carbonic anhydrases and mucosal vanilloid receptors help mediate the hyperemic response to luminal CO2 in rat duodenum GASTROENTEROLOGY 131 (1): 142-152 JUL 2006 Pomarnacka E (Pomarnacka, Elzbieta), Bednarski PJ (Bednarski, Patrick J.), Reszka P (Reszka, Przemyslaw), Dziemidowicz-Borys E (Dziemidowicz-Borys, Ewa), Bienczak A (Bienczak, Andrzej), Werel W (Werel, Wladyslaw), Halasa R (Halasa, Rafal) Synthesis and biological activity of new 2-amino-8-chloro-5,5-dioxo[1,2,4]triazolo[2,3-b][1,4,2]benzodithiazines EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY 41 (5): 633-639 MAY 2006 Poulsen SA, Bornaghi LF Fragment-based drug discovery of carbonic anhydrase II inhibitors by dynamic combinatorial chemistry utilizing alkene cross metathesis BIOORGANIC & MEDICINAL CHEMISTRY 14 (10): 3275-3284 MAY 15 2006 Guler OO (Guler, O. Ozensoy)1, Arslan O (Arslan, O.)1, Kockar F (Kockar, F.)2 Differential in vitro inhibitory effects of anticancer drugs on tumor-associated carbonic anhydrase isozymes CA IX and CA XII METHODS AND FINDINGS IN EXPERIMENTAL AND CLINICAL PHARMACOLOGY Volume: 30 Issue: 5 Pages: 335-340 Published: JUN 2008 Adamski JK, Estlin EJ, Makin GWJ The cellular adaptations to hypoxia as novel therapeutic targets in childhood cancer CANCER TREATMENT REVIEWS Volume: 34 Issue: 3 Pages: 231-246 Published: MAY 2008 Parkkila S (Parkkila, Seppo)1,2,3 Significance of pH regulation and carbonic anhydrases in tumour progression and implications for diagnostic and therapeutic approaches BJU INTERNATIONAL Volume: 101 Pages: 16-21 Supplement: Suppl. 4 Published: JUN 2008 Vu H, Quinn RJ Direct screening of natural product extracts using mass spectrometry JOURNAL OF BIOMOLECULAR SCREENING Volume: 13 Issue: 4 Pages: 265-275 Published: APR 2008 Hofmeister V, Schrama D, Becker JC Anti-cancer therapies targeting the tumor stroma CANCER IMMUNOLOGY IMMUNOTHERAPY Volume: 57 Issue: 1 Pages: 1-17 Published: JAN 2008 Sharma BK (Sharma, Brij Kishore)1, Pilania P (Pilania, Pradeep)1, Singh P (Singh, Prithvi)1, Sharma S (Sharma, Susheela)2, Prabhakar YS (Prabhakar, Yenamandra S.)3 CP-MLR directed QSAR study of carbonic anhydrase inhibitors: sulfonamide and sulfamate inhibitors CENTRAL EUROPEAN JOURNAL OF CHEMISTRY Volume: 7 Issue: 4 Pages: 909-922 Published: DEC 2009 Robertson L, Hartley RC Synthesis of N-arylpyridinium salts bearing a nitrone spin trap as potential mitochondria-targeted antioxidants TETRAHEDRON Volume: 65 Issue: 27 Pages: 5284-5292 Published: JUL 4 2009 Abdel-Hamid MK (Abdel-Hamid, Mohammed K.)1, Abdel-Hafez AA (Abdel-Hafez, Atef A.)1, El-Koussi NA (El-Koussi, Nawal A.)1, Mahfouz NM (Mahfouz, Nadia M.)1 Quantitative structure-activity relationship (QSAR) studies on a series of 1,3,4-thiadiazole-2-thione derivatives as tumor-associated carbonic anhydrase IX inhibitors JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY Volume: 24 Issue: 3 Pages: 722-729 Published: 2009 Akula NVMK (Akula, N. V. Murali Krishna)1, Kumar S (Kumar, Surendra)1, Singh V (Singh, Vineet)1, Tiwari M (Tiwari, Meena)1 Homology modeling and QSAR analysis of 1,3,4-thiadiazole and 1,3,4-triazole derivatives as carbonic anhydrase inhibitors INDIAN JOURNAL OF BIOCHEMISTRY & BIOPHYSICS Volume: 47 Issue: 4 Pages: 234-242 Published: AUG 2010 Apte Sandeep; Chin Frederick T.; Graves Edward E. Molecular Imaging of Hypoxia: Strategies for Probe Design and Application CURRENT ORGANIC SYNTHESIS Volume: 8 Issue: 4 Pages: 593-603 Published: AUG 2011 Kasimogullari, R (Kasimogullari, Rahmi)1; Bulbul, M (Bulbul, Metin)1; Mert, S (Mert, Samet)1; Guleryuz, H (Guleryuz, Hulya)1 Synthesis of 5-amino-1,3,4-thiadiazole-2-sulphonamide derivatives and their inhibition effects on human carbonic anhydrase isozymes JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY Volume: 26 Issue: 2 Pages: 231-237 DOI: 10.3109/14756366.2010.491795 Published: APR 2011 Mohamed, N.A., Anwar, M.M., El-Serwy, W.S., Elsherbiny, M Synthesis and cytotoxicity of novel Hexahydroquinoline-benzenesulfonamide derivatives Der Pharma Chemica 4 (5) , pp. 2055-2067 , 2012 Aggarwal, Mayank; McKenna, Robert Update on carbonic anhydrase inhibitors: a patent review (2008-2011) EXPERT OPINION ON THERAPEUTIC PATENTS Volume: 22 Issue: 8 Pages: 903-915 DOI: 10.1517/13543776.2012.707646 Published: AUG 2012 Liu, CM (Liu, Chia-Ming)[ 2,3 ] ; Lin, YM (Lin, Yueh-Min)[ 4,5 ] ; Yeh, KT (Yeh, Kun-Tu)[ 4,6 ] ; Chen, MK (Chen, Mu-Kuan)[ 6,7 ] ; Chang, JH (Chang, Jer-Hwa)[ 8,9 ] ; Chen, CJ (Chen, Chih-Jung)[ 4,5,10 ] ; Chou, MY (Chou, Ming-Yung)[ 2,3 ] ; Yang, SF (Yang, Shun-Fa)[ 10,11 ] ; Chien, MH (Chien, Ming-Hsien)[ 1,8 ] Expression of carbonic anhydrases I/II and the correlation to clinical aspects of oral squamous cell carcinoma analyzed using tissue microarray JOURNAL OF ORAL PATHOLOGY & MEDICINE Volume: 41 Issue: 7 Pages: 533-539 DOI: 10.1111/j.1600-0714.2012.01135.x Published: AUG 2012 Doss, M (Doss, Mohan)[ 1 ] ; Kolb, HC (Kolb, Hartmuth C.)[ 2 ] ; Walsh, JC (Walsh, Joseph C.)[ 2 ] ; Mocharla, VP (Mocharla, Vani P.)[ 2 ] ; Zhu, ZH (Zhu, Zhihong)[ 3 ] ; Haka, M (Haka, Michael)[ 3 ] ; Alpaugh, RK (Alpaugh, R. Katherine)[ 4 ] ; Chen, DYT (Chen, David Y. T.)[ 5 ] ; Yu, JQ Biodistribution and Radiation Dosimetry of the Carbonic Anhydrase IX Imaging Agent [(18) F]VM4-037 Determined from PET/CT Scans in Healthy Volunteers MOLECULAR IMAGING AND BIOLOGY Volume: 16 Issue: 5 Pages: 739-746, 2014 Tafreshi, NK (Tafreshi, Narges K.)[ 1 ] ; Lloyd, MC (Lloyd, Mark C.)[ 2 ] ; Bui, MM (Bui, Marilyn M.)[ 2,3 ] ; Gillies, RJ (Gillies, Robert J.)[ 1 ] ; Morse, DL Carbonic Anhydrase IX as an Imaging and Therapeutic Target for Tumors and Metastases Edited by:Frost, SC; McKenna, R CARBONIC ANHYDRASE: MECHANISM, REGULATION, LINKS TO DISEASE, AND INDUSTRIAL APPLICATIONS Book Series: Subcellular Biochemistry Volume: 75 Pages: 221-254, 2014 Iqbal, S (Iqbal, Shoaib)[ 1 ] ; Nisar-ur-Rahman (Nisar-ur-Rahman)[ 1 ] ; Iqbal, J A capillary electrophoresis-based enzyme assay for kinetics and inhibition studies of carbonic anhydrase ANALYTICAL BIOCHEMISTRY Volume: 444 Pages: 16-21, 2014 Mahon, BP (Mahon, Brian P.)[ 1 ] ; Pinard, MA (Pinard, Melissa A.)[ 1 ] ; McKenna, R Targeting Carbonic Anhydrase IX Activity and Expression MOLECULES Volume: 20 Issue: 2 Pages: 2323-2348, 2015 MCINTYRE, Alan - HARRIS, Adrian L. The Role of pH Regulation in Cancer Progression. In METABOLISM IN CANCER. ISSN 0080-0015, 2016, vol. 207, no., pp. 93-134. JUOZAPAITIENE, Vaida - BARTKUTE, Brigita - MICHAILOVIENE, Vilma - ZAKSAUSKAS, Audrius - BARANAUSKIENE, Lina - SATKUNE, Sandra - MATULIS, Daumantas. Purification, enzymatic activity and inhibitor discovery for recombinant human carbonic anhydrase XIV. In JOURNAL OF BIOTECHNOLOGY. ISSN 0168-1656, 2016, vol. 240, no., pp. 31-42. JUN, So-Young - KIM, Sung Ho - KANTH, Bashista Kumar - LEE, Jinwon - PACK, Seung Pil. Expression and characterization of a codon-optimized alkaline-stable carbonic anhydrase from Aliivibrio salmonicida for CO2 sequestration applications. In BIOPROCESS AND BIOSYSTEMS ENGINEERING. ISSN 1615-7591, 2017, vol. 40, no. 3, pp. 413-421. MILITE, Ciro - AMENDOLA, Giorgio - NOCENTINI, Alessio - BUA, Silvia - CIPRIANO, Alessandra - BARRESI, Elisabetta - FEOLI, Alessandra - NOVELLINO, Ettore - DA SETTIMO, Federico - SUPURAN, Claudiu T. - CASTELLANO, Sabrina - COSCONATI, Sandro - TALIANI, Sabrina. Novel 2-substituted-benzimidazole-6-sulfonamides as carbonic anhydrase inhibitors: synthesis, biological evaluation against isoforms I, II, IX and XII and molecular docking studies. In JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY. ISSN 1475-6366, 2019, vol. 34, no. 1, pp. 1697-1710. EL KHARRAT, Salem - LAURENT, Philippe - BOITEAU, Laurent - BLANCOU, Hubert. Novel Synthesis of Substituted 2-Trifluoromethyl and 2-Perfluoroalkyl N-Arylpyridinium Compounds-Mechanistic Insights. In MOLECULES, 2019, vol. 24, no. 12, pp. NEMR, M.T.M. - ABOULMAGD, A.M. - HASSAN, H.M. - HAMED, A.A. - HAMED, M.I.A. - ELSAADI, M.T. Design, synthesis and mechanistic study of new benzenesulfonamide derivatives as anticancer and antimicrobial agents via carbonic anhydrase IX inhibition. In RSC ADVANCES. AUG 10 2021, vol. 11, no. 42, p. 26241-26257. Dostupné na: https://doi.org/10.1039/d1ra05277b. TUGRAK, M. - GUL, H.I. - SAKAGAMI, H. - KAYA, R. - GULCIN, I. Synthesis and biological evaluation of new pyrazolebenzene-sulphonamides as potential anticancer agents and hCA I and II inhibitors. In TURKISH JOURNAL OF CHEMISTRY. ISSN 1300-0527, 2021, vol. 45, no. 3, p. 528-+. Dostupné na: https://doi.org/10.3906/kim-2009-37. KORKMAZ, Isil Nihan - GULLER, Pinar - KALIN, Ramazan - OZTEKIN, Aykut - OZDEMIR, Hasan. iIn vitro/i Inhibition Profiles and Molecular Docking Analysis of Benzohydrazide Derivatives on Red Blood Cell Carbonic Anhydrases Isozymes. In CURRENT COMPUTER-AIDED DRUG DESIGN. ISSN 1573-4099, 2022, vol. 18, no. 5, p. 381-392. Dostupné na: https://doi.org/10.2174/1573409918666220818114505. Kategória ADCA - Vedecké práce v zahraničných karentovaných časopisoch impaktovaných Kategória (od 2022) V3 - Vedecký výstup publikačnej činnosti z časopisu Typ výstupu článok Rok vykazovania 2004 
článok
rok CC IF IF Q (best) JCR Av Jour IF Perc SJR SJR Q (best) CiteScore A rok vydania rok metriky IF IF Q (best) SJR SJR Q (best) 2004 2003 2.182
Počet záznamov: 1